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Cat. No. Product Name Target Signaling Pathways
T31716L Etidocaine

Others Others
Etidocaine 是一种氨基酸酰胺,用作局部麻醉剂,具有快速起效和长效特性。
T31716 Etidocaine Hydrochloride

W-19053,Duranest,W19053,W 19053

Sodium Channel Membrane transporter/Ion channel
Etidocaine Hydrochloride (W19053) 是一种长效麻醉剂和电压门控钠通道阻滞剂。
T0901 Chlorobutanol

Chlortran,Chloretone,YM-57158,三氯叔丁醇,Chlorbutol,Chloreton

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Chlorobutanol (Chlortran) 是一种药物防腐剂,对多种革兰氏阳性和革兰氏阴性细菌以及几种霉菌孢子和真菌具有抗性。它广泛用于食品和化妆品工业,有促进安定、睡眠的作用。
T0030 Bupivacaine hydrochloride

Vivacaine,Bupivacaine HCl,盐酸布比卡因

Sodium Channel Membrane transporter/Ion channel
Bupivacaine hydrochloride (Vivacaine) 是NMDA 受体抑制剂,可用于慢性疼痛的研究。它可阻断钠、L-钙和钾通道,还阻断SCN5A 通道,IC50为 69.5 μM。
T22425 Sevoflurane

七氟烷,Fluoromethyl

5-HT Receptor GPCR/G Protein; Neuroscience
Sevoflurane (Fluoromethyl) 是一种 5-HT3 受体的非竞争性抑制剂,是一种低溶性吸入麻醉剂。
T2387 Glycopyrrolate

Gastrodyn,Glycopyrronium bromide,Robinul,Glycopyrrolate bromide,格隆溴铵

AChR Neuroscience
Glycopyrrolate (Glycopyrrolate bromide) 是一种毒蕈碱拮抗剂,在某些胃肠道疾病中用作解痉剂,并与某些麻醉剂一起减少唾液分泌。
T34072 Pipotiazine

19366 RP,Pipotiazina,Pipotiazinum,Piportil L4,Pipothiazine

Pipotiazine has less sedating and a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetics among the different phenothiazine derivatives. However, it produces a high incidence of extra pyramidal reactions. I
T37670 CAY10568

Most local anesthetics act by abolishing voltage gated sodium channel currents indiscriminately in all populations of neurons. Selective analgesia through TRPV1-mediated entry of a cationic lidocaine derivative, QX314, was recently reported. CAY10568 is a physically smaller, less hydrophobic version of QX314 designed to be even more permeable to TRPV1 ion channel when activated by agonists such as capsaicin and N-oleoyl dopamine. CAY10568 when given in combination with suitable TRPV1 agonists sh...
T60469 Chloroprocaine

Chloroprocaine (2-Chloroprocaine) 是一种有效的Na,K-ATPase 酶活性抑制剂(IC50 = 13 mM)。Chloroprocaine 是一种阻滞外周神经的局部麻醉剂。

化合物

Etidocaine
Cat.No: T31716L
Synonym:
Target: Others
Etidocaine Hydrochloride
Cat.No: T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
Chlorobutanol
Cat.No: T0901
Synonym: Chlortran,Chloretone,YM-57158,三氯叔丁醇,Chlorbutol,Chloreton
Target: Antibacterial, Antibiotic, Antifungal
Bupivacaine hydrochloride
Cat.No: T0030
Synonym: Vivacaine,Bupivacaine HCl,盐酸布比卡因
Target: Sodium Channel
Sevoflurane
Cat.No: T22425
Synonym: 七氟烷,Fluoromethyl
Target: 5-HT Receptor
Glycopyrrolate
Cat.No: T2387
Synonym: Gastrodyn,Glycopyrronium bromide,Robinul,Glycopyrrolate bromide,格隆溴铵
Target: AChR
Pipotiazine
Cat.No: T34072
Synonym: 19366 RP,Pipotiazina,Pipotiazinum,Piportil L4,Pipothiazine
Target:
CAY10568
Cat.No: T37670
Synonym:
Target:
Chloroprocaine
Cat.No: T60469
Synonym:
Target:
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