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Search Results for " alpha 1-adrenoceptor "

16

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T3046	BMY 7378 dihydrochloride BMY7378 HCl	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	BMY 7378 dihydrochloride (BMY7378 HCl) 是选择性 α1D 肾上腺素受体拮抗剂，也是5-HT1A 受体部分激动剂。它同表达克隆大鼠 α1D-AR 的膜结合的亲和力 (Ki=2 nM) 是同克隆大鼠 α1A-AR (Ki=800 nM) 或仓鼠 α1B-AR (Ki=600 nM) 结合的亲和力的100 以上。
T26923	Bunazosin Hydrochloride E 1015,盐酸布那唑嗪,E643,E-1015,E-643,E 643	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Bunazosin Hydrochloride (E 1015) 是一种 α(1)-adrenoceptor 拮抗剂，用作全身性抗高血压药和降眼压药。
T10003	α1 adrenoceptor-MO-1	Others	Others
	α1 adrenoceptor-MO-1（S 对映体）对α1肾上腺素受体具有亲和力，具有抗α-肾上腺素能和镇痛作用。α1 adrenoceptor-MO-1比R 对映体更具活性。
T10364	Arbutamine GP 21213	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Arbutamine (GP 21213) 是一种新型非选择性β-肾上腺素受体激动剂，具有α-1-拟交感神经活性。Arbutamine 促进心脏应激，增加心率、心脏收缩力。Arbutamine 可用于研究心脏应激和冠状动脉疾病。
T22232	Alfuzosin
	Alfuzosin 是选择性和竞争性的α1肾上腺素受体拮抗剂，可用于良性前列腺增生（BPH）的研究。
T28789	SKF 89748 SKF89748,SKF0-89748
	SKF 89748 is an agonists of alpha 1-adrenoceptor.
T68772	Ocoteine
	Ocoteine is an alpha 1-adrenoceptor antagonist.
T68636	Indanidine hydrochloride
	Indanidine hydrochloride is an alpha 1 adrenoceptor agonist.
T26507	Abanoquil
	Abanoquil is an antagonist of alpha-1 adrenoceptor.
T71104	HSR-175 HCl
	HSR-175 HCl is an alpha 1-adrenoceptor antagonist.
T71366	HV-723 fumarate
	HV-723 fumarate is an alpha-1 adrenoceptor antagonist.
T70537	DC 015
	DC 015 is a novel potent and selective alpha 1-adrenoceptor antagonist.
T69075	Dicentrine HCl
	Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.
T25333	Dilevalol Dilevalolum
	Dilevalol, the RR-stereoisomer of labetalol, is a non-cardioselective beta-adrenoceptor antagonist with substantial partial beta 2-agonist and negligible alpha 1-blocking activity.
T21787	B-HT 933 dihydrochloride
	Azepexole (B-HT 933) dihydrochloride 是一种有效的选择性α 2肾上腺素受体激动剂，对 α2A-、α2B- 和 α2C- 肾上腺素受体亚型的 pKi 分别为 8.3、7.6 和 7.5。Azepexole dihydrochloride 引起浓度依赖性的蠕动收缩抑制，IC50值为 78.72 nM。
T37794	Rec 15/2615 (hydrochloride)
	Rec 15/2615 is an antagonist of α1B-adrenergic receptors (α1B-ARs; Ki = 0.45 nM for the recombinant human receptor).1 It selectively inhibits α1B-ARs over α1A-, α1D-, and α1L-ARs (Kis = 7.59, 10.23, and 49 nM, respectively). Rec 15/2615 inhibits norepinephrine-induced contractions of isolated rabbit prostate and urethral strips (Kis = 100 and 316.2 nM, respectively), as well as reduces norepinephrine-induced contractions of chloroethylclonidine-precontracted isolated rabbit aortic rings (Ki = 50...

化合物

BMY 7378 dihydrochloride

Cat.No: T3046

Synonym: BMY7378 HCl

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Bunazosin Hydrochloride

Cat.No: T26923

Synonym: E 1015,盐酸布那唑嗪,E643,E-1015,E-643,E 643

Target: Adrenergic Receptor

α1 adrenoceptor-MO-1

Cat.No: T10003

Target: Others

Cat.No: T10364

Synonym: GP 21213

Target: Adrenergic Receptor

Cat.No: T22232

Cat.No: T28789

Synonym: SKF89748,SKF0-89748

Cat.No: T68772

Indanidine hydrochloride

Cat.No: T68636

Cat.No: T26507

Cat.No: T71104

HV-723 fumarate

Cat.No: T71366

Cat.No: T70537

Cat.No: T69075

Cat.No: T25333

Synonym: Dilevalolum

B-HT 933 dihydrochloride

Cat.No: T21787

Rec 15/2615 (hydrochloride)

Cat.No: T37794

Cat. No.	Product Name	Target	Signaling Pathways
TN3507	beta-Yohimbine	Adrenergic Receptor; Antifection	GPCR/G Protein; Microbiology/Virology; Neuroscience
	Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor blocking activities, it has cardiovascular effects. Beta-Yohimbine has anti-plasmodial and anti-mal
TN5061	Stephanine	Adrenergic Receptor; Antifection	GPCR/G Protein; Microbiology/Virology; Neuroscience
	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. Stephanine shows significant antiplasmodial activities with IC(50) ranged from 1.2 uM to 52.3 uM. Stephanine and crebanine have high inhibitory activity against gram-positive animal pathogenic bacteria, with MIC values of 0.078-0.312g/l, but low inhibitory activity against gram-negative animal pathogenic bacteria, they also inhibit...

天然产物

Cat.No: TN3507

Target: Adrenergic Receptor, Antifection

Cat.No: TN5061

Target: Adrenergic Receptor, Antifection

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