Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11005 |
Desmethyl Celecoxib
|
COX | Immunology/Inflammation; Neuroscience |
Desmethyl Celecoxib 是一种选择性的环氧化酶 2 (COX-2) 抑制剂,IC50为 32 nM,具有抗炎活性。 | |||
T22632 |
TASIN-1
1-[(4-methoxyphenyl)sulfonyl]-4'-methyl-4,1'-bipiperidine,塔辛-1 |
APC | Cell Cycle/Checkpoint |
TASIN-1 是截短的APC 基因(结肠腺瘤样息肉基因)选择性抑制剂,可以抑制胆固醇生物合成并发挥细胞毒性作用。它是一种预防和干预APC 突变型结直肠癌的潜在治疗策略。 | |||
T32026 |
GYKI-13324
GYKI 13324,GYKI13324 |
||
GYKI-13324 is bifunctional nitrosoureido derivative and alkylating agent. GYKI-13324 was studied on human colorectal tumor xenograft lines. Given orally in single or multiple daily doses, GYKI-13324 produced long-term or total regression of adenomatous, b | |||
T81876 |
MAIT-203
|
||
MAIT-203为环戊丙氨酸衍生的拟肽,专一抑制APC和Asef (RhoGEF4)的相互作用,不影响APC-Sam68或APC-striatin。该化合物与APC-ARM结合紧密,Ki值为0.015 μM,Kd值为0.036 μM,并有效抑制结直肠癌细胞的迁移与侵袭。 |