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Cat. No. Product Name Target Signaling Pathways
T2154 MG-132

Z-LLL-al,Z-Leu-Leu-Leu-CHO

Apoptosis; Proteasome; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
MG-132 (Z-Leu-Leu-Leu-al) 是一种 26S 蛋白酶体抑制剂 (IC50=100 nM),具有细胞渗透性、可逆性。MG-132 可作为自噬激活剂,可诱导凋亡。
T78640 Z-LLF-CHO

Z-Leu-Leu-Phe-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-LLF-CHOZ-Leu-Leu-Phe-CHO)为垂体多催化蛋白酶复合物所具有的胰凝乳蛋白酶样活性提供有效抑制,具有Ki值为460 nM。此外,Z-LLF-CHO同样作为NF-κB核转位的抑制剂。
T17281 Z-Ile-Leu-aldehyde

Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII

Others Others
Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.
T80735 Z-Gly-Pro-Phe-Leu-CHO

Z-GPFL-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-Gly-Pro-Phe-Leu-CHOZ-GPFL-CHO)是一种具有高选择性和高效率的四肽醛类蛋白酶体抑制剂,优先抑制支链氨基酸(Ki为1.5 µM),对小中性氨基酸的Ki值为2.3 µM,胰凝乳蛋白酶样活性的Ki值为40.5 µM,对肽基-谷氨酰肽水解活性的IC50为3.1 µM。

化合物

MG-132
Cat.No: T2154
Synonym: Z-LLL-al,Z-Leu-Leu-Leu-CHO
Target: Apoptosis, Proteasome, Autophagy
Z-LLF-CHO
Cat.No: T78640
Synonym: Z-Leu-Leu-Phe-CHO
Target: Proteasome
Z-Ile-Leu-aldehyde
Cat.No: T17281
Synonym: Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII
Target: Others
Z-Gly-Pro-Phe-Leu-CHO
Cat.No: T80735
Synonym: Z-GPFL-CHO
Target: Proteasome
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