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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T35723 GRK-IN-1

4-Amino-5-(bromomethyl)-2-methylpyrimidine is a heterocyclic building block.1,2 It has been used in the synthesis of vitamin B1 analogs and thiaminephosphoric acid esters. |1. Abblard, J., Cronenberger, L., and Pacheco, H. Synthesis of the analogs of vitamin B1. Chim. Ther. 8(1), 98-110 (1973).|2. Leichssenring, G., and Joachim, S. The synthesis of thiaminephosphoric acid esters. Chem. Ber. 95, 767-772 (1962).
T35983 Carotenoid Mixture

Carotenoid mixture is a mixture of carotenoids that contains the antioxidative and anti-inflammatory carotenoid capsanthin and the antioxidative vitamin A precursor β-carotene , as well as additional carotenoids and carotenoid esters.1,2,3,4 1.Kim, J.S., Lee, W.M., Rhee, H.C., et al.Red paprika (Capsicum annuum L.) and its main carotenoids, capsanthin and β-carotene, prevent hydrogen peroxide-induced inhibition of gap-junction intercellular communicationChem. Biol. Interact.254146-155(2016) 2.Na...

化合物

GRK-IN-1
Cat.No: T35723
Synonym:
Target:
Carotenoid Mixture
Cat.No: T35983
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1116 Biotin

Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H

Biotin (Vitamin H) 是一种水溶性B族维生素,是细胞生长、脂肪酸产生以及脂肪和氨基酸代谢所必需的。
T1311 4-aminobenzoic acid

PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸

Endogenous Metabolite Metabolism
4-aminobenzoic acid (para-Aminobenzoic acid) 是一种具有紫外线吸收和抗纤维化特性的有机酸。当暴露在光线下时,4-aminobenzoic acid 吸收紫外线并通过光化学反应释放多余的能量,这可能会对DNA造成损害。4-aminobenzoic acid 还可以增加组织水平的摄氧量,并可能增强单胺氧化酶(MAO)活性以促进血清素的降解,过量可能导致纤维化变化。
T0809 Dicoumarol

Dicumarol,双羟香豆素,双香豆素

Dehydrogenase; NADPH; PDK Metabolism; PI3K/Akt/mTOR signaling
Dicoumarol (Dicumarol) 是一种 NAD(P)H: 醌氧化还原酶 1 和PDK1的抑制剂,它们的IC50值分别为 0.37 和 19.42 μM。

天然产物

Biotin
Cat.No: T1116
Synonym: Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H
Target:
4-aminobenzoic acid
Cat.No: T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸
Target: Endogenous Metabolite
Dicoumarol
Cat.No: T0809
Synonym: Dicumarol,双羟香豆素,双香豆素
Target: Dehydrogenase, NADPH, PDK
TargetMol Loading
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