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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T37406 Apovincaminic acid hydrochloride salt

Apovincaminic acid hydrochloride salt, the primary active metabolite of Vinpocetine (VP), is orally active and has the ability to penetrate the brain. It demonstrates a neuroprotective mechanism of action [1][2].

化合物

Apovincaminic acid hydrochloride salt
Cat.No: T37406
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0167 Vinpocetine

长春西丁,RGH-4405,长春西汀,Ethyl apovincaminate

IκB/IKK; NF-κB; Sodium Channel; PDE Membrane transporter/Ion channel; Metabolism; NF-κB
Vinpocetine (RGH-4405) 是一种长春花生物碱衍生物,是阻断 Na+通道的阻断剂。Vinpocetine 抑制IKK 的IC50为 17.17 μM。Vinpocetine 也是PDE 抑制剂,并通过直接靶向IKK 抑制NF-κB 依赖性炎症反应,已被广泛用于研究脑血管疾病。
T21047 Apovincamine

cis-Apovincamine

Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity.

天然产物

Vinpocetine
Cat.No: T0167
Synonym: 长春西丁,RGH-4405,长春西汀,Ethyl apovincaminate
Target: IκB/IKK, NF-κB, Sodium Channel, PDE
Apovincamine
Cat.No: T21047
Synonym: cis-Apovincamine
Target:
TargetMol Loading
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