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Search Results for " thyrotropin "

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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T80985	Thyrotropin Pretiron,TSH
	Thyrotropin (TSH)为促甲状腺激素，由垂体前叶的促甲状腺细胞分泌，主要功能是调节甲状腺的内分泌活动。
T7407	Thyrotropin-Releasing Hormone (TRH), Free Acid TRH-OH	Others	Others
	Thyrotropin-Releasing Hormone (TRH), Free Acid (TRH-OH) 是一种促甲状腺激素释放激素的生理代谢产物。
T6956L	Protirelin Acetate(24305-27-9 free base) Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate	Thyroid hormone receptor(THR)	Endocrinology/Hormones
	Protirelin Acetate(24305-27-9 free base) (Thyroliberin Acetate) 是一种三肽，可刺激促甲状腺素和催乳素的释放。
T34869	Thyrotropin-releasing hormone, deamido- Deamido-trh,Pyroglutamyl-histidyl-proline,Trh-OH,Trh, deamido-,Pglu-his-pro
	Thyrotropin-releasing hormone, deamido- is a biochemical.
T34206	Pyroglutaminyl-seryl-leucinamide Thyrotropin releasing hormone-AN,Trh-AN,Pyr-ser-leu-NH2
	Pyroglutaminyl-seryl-leucinamide is a bioactive chemical.
T12073	ML-109	TSH Receptor	GPCR/G Protein
	ML-109 是一种促甲状腺激素受体的有效激动剂，EC50值为 40 nM。
T12192	NCGC00229600	Others; TSH Receptor	GPCR/G Protein; Others
	NCGC00229600 是促甲状腺激素受体 (TSHR) 的变构反向激动剂。 NCGC00229600 抑制 TSH 和刺激 TSHR 的内源性激活抗体，可用于格雷夫斯病的研究。
T5383	D3-βArr NCGC00379308	TSH Receptor	GPCR/G Protein
	D3-βArr (NCGC00379308) 是一种促甲状腺激素受体正变构调节剂，通过直接激活促甲状腺激素受体启动 β-Arr 1 的易位，EC50为 11.6 μM。它还可增强促甲状腺激素介导的体外成骨细胞分化。
TP1022	Protirelin Acetate TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林	Thyroid hormone receptor(THR); Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Protirelin Acetate (TRH Acetate) 是高度保守的神经肽，具有促甲状腺激素水平的激素控制作用，及神经调节的能力。
T33824	Orotirelin CG 3509,Orotireline	Others	Others
	Orotirelin(CG 3509) 是促甲状腺激素释放激素类似物，可逆转了戊巴比妥诱导的睡眠时间。Orotirelin 可能对局灶性脑缺血的动物有益。
T29087	VA-K-14 hydrochloride VAK14 Hydrochloride,VA K 14 HCl,VA-K-14 HCl,VAK14 HCl	TSH Receptor	GPCR/G Protein
	VA-K-14 hydrochloride（VAK14 HCl）是一种选择性促甲状腺激素受体 (TSHR) 拮抗剂 (IC50= 12.3 μM)，对GD患者血清和单克隆刺激TSHR抗体对TSHR的刺激有抑制作用，可消除 TSHR 信号传导。
T13216	TSHR antagonist S37	TSH Receptor	GPCR/G Protein
	TSHR antagonist S37 是促甲状腺激素受体 (TSHR) 的选择性和竞争性拮抗剂。
T34399	Rovatirelin KPS-0373,S0373,S-0373,S 0373	AChE	Neuroscience
	Rovatirelin (S-0373) 是一种新合成的促甲状腺激素释放激素（TRH）类似物，通过乙酰胆碱和多巴胺神经传递改善胞嘧啶阿拉伯糖苷诱导的脊髓小脑变性大鼠模型的运动功能障碍。
T13072	Taltirelin acetate TA-0910 acetate	Thyroid hormone receptor(THR)	Endocrinology/Hormones
	Taltirelin acetate (TA-0910 acetate) 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM)，能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) ，其EC50值为 36 nM。
T33480	Montirelin NS 3,Montirelinum,CNK 602A,CNK-603
	Montirelin is an analog of thyrotropin-releasing hormone.
T34923	TRH tartrate
	TRH tartrate is a thyrotropin-releasing hormone.
T32317	Jtp 2942 Jtp2942,Jtp-2942
	Jtp 2942 is a new thyrotropin-releasing hormone analog.
T31553	DN 1417 DN1417,DN-1417
	DN 1417 is an analog of thyrotropin releasing hormone.
T77258	Trh-gly
	Trh-gly (TRH-glycine) 是促甲状腺素 (TSH) 释放激素 (TRH) 的前体，可释放促甲状腺素和催乳素。
T16972	TA 0910 acid-type	Others	Others
	TA 0910 acid-type is a metabolite of TA 0910. TA-0910 is a metabolically stable analog of thyrotropin-releasing hormone.
TP2201	TRH Precursor Peptide	Others	Others
	Thyrotropin Releasing Hormone Precursor Peptide
T76494	[Phe2]-TRH
	[Phe2]-TRH 是一种促甲状腺激素释放激素类似物，与 Leu5-脑啡肽具有构象相似性。
T13217	TSHR antagonist S37a	Others	Others
	TSHR antagonist S37a is a selective antagonist of thyrotropin receptor (TSHR), with potential for the treatment of Graves' orbitopathy.
T76496	Prepro-TRH-(160-169)
	Prepro-TRH-(160-169)，作为促甲状腺激素释放激素原 (pro-TRH) 的连接肽之一，具有增强TRH诱导的促甲状腺激素 (TSH) 释放的功能。
T38226	TSHR antagonist S37b
	TSHR antagonist S37b, the less potent enantiomer of TSHR antagonist S37a, exhibits minimal efficacy in inhibiting the thyrotropin receptor (TSHR). It is utilized in thyroid function research[1].
T33438	MK771 MK-771,MK 771
	MK771 is a therapeutic agent and an analog of the Thyrotropin Releasing Hormone (TRH). TRH and its analogs may be useful in combating some of the withdrawal symptoms in opiate-dependent subjects.
T70365	JTP-4819
	JTP-4819 is a potent and selective prolyl endopeptidase (PEP) inhibitor with potential for treating Alzheimer's disease. At nanomolar concentration, JTP-4819 inhibited the degradation of substance P, arginine-vasopressin, and thyrotropin-releasing hormone by PEP in supernatants of the rat cerebral cortex and hippocampus. Repeated administration of JTP-4819 reversed the aging-induced decrease in brain substance P-like and thyrotropin-releasing hormone-like immunoreactivity, suggesting that this d...
T7590	Taltirelin TA-0910,他替瑞林	Thyroid hormone receptor(THR)	Endocrinology/Hormones
	Taltirelin (TA-0910) 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM)，能够刺激细胞溶质 Ca2+浓度增加 (Ca2+释放) (EC50:36 nM)。
TP2011	JKC363 JKC 363
	Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 0.5 and 44.9 nM at MC4 and MC3 respectively) that antagonizes the effects of α-MSH. Suppresses thyrotropin-releasing hormone (TRH) release, attenuates food intake and reduces forma
T76493	(Glu2)-TRH
	(Glu2)-TRH 是一种代谢稳定的 Thyrotropin-releasing hormone(TRH) 类似物，是小鼠大脑中 TRH 胆碱能作用的负调节剂。(Glu2)-TRH 显着减弱 TRH 诱导的海马细胞外乙酰胆碱释放。(Glu2)-TRH 不被甲状腺解放酶代谢。(Glu2)-TRH 在中枢神经系统中表现出神经保护、抗抑郁、抗惊厥作用。
T36383	L-Thyroxine-13C9,15N L-Thyroxine-13C9,15N
	L-Thyroxine-13C9,15N is intended for use as an internal standard for the quantification of L-thyroxine by GC- or LC-MS. L-Thyroxine is a synthetic form of the thyroid hormone thyroxine. In vivo, L-thyroxine (0.9 and 2.7 μg) inhibits synthesis and release of thyrotropin induced by thyrotropin-releasing hormone from the anterior pituitary in mice. It also reverses decreases in levels of circulating thymic serum factor (FTS) and the number of T rosette-forming cells in an old age-induced mouse mode...
TMIH-0550	Taltirelin-13C-d3
	Taltirelin-13C-d3 是 Taltirelin 的 13C 和氘代化合物。Taltirelin 的 CAS 号为 103300-74-9。Taltirelin 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM)，能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) (EC50:36 nM)。

化合物

Cat.No: T80985

Synonym: Pretiron,TSH

Thyrotropin-Releasing Hormone (TRH), Free Acid

Cat.No: T7407

Synonym: TRH-OH

Target: Others

Protirelin Acetate(24305-27-9 free base)

Cat.No: T6956L

Synonym: Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate

Target: Thyroid hormone receptor(THR)

Thyrotropin-releasing hormone, deamido-

Cat.No: T34869

Synonym: Deamido-trh,Pyroglutamyl-histidyl-proline,Trh-OH,Trh, deamido-,Pglu-his-pro

Pyroglutaminyl-seryl-leucinamide

Cat.No: T34206

Synonym: Thyrotropin releasing hormone-AN,Trh-AN,Pyr-ser-leu-NH2

Cat.No: T12073

Target: TSH Receptor

Cat.No: T12192

Target: Others, TSH Receptor

Cat.No: T5383

Synonym: NCGC00379308

Target: TSH Receptor

Protirelin Acetate

Cat.No: TP1022

Synonym: TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林

Target: Thyroid hormone receptor(THR), Endogenous Metabolite

Cat.No: T33824

Synonym: CG 3509,Orotireline

Target: Others

VA-K-14 hydrochloride

Cat.No: T29087

Synonym: VAK14 Hydrochloride,VA K 14 HCl,VA-K-14 HCl,VAK14 HCl

Target: TSH Receptor

TSHR antagonist S37

Cat.No: T13216

Target: TSH Receptor

Cat.No: T34399

Synonym: KPS-0373,S0373,S-0373,S 0373

Target: AChE

Taltirelin acetate

Cat.No: T13072

Synonym: TA-0910 acetate

Target: Thyroid hormone receptor(THR)

Cat.No: T33480

Synonym: NS 3,Montirelinum,CNK 602A,CNK-603

Cat.No: T34923

Cat.No: T32317

Synonym: Jtp2942,Jtp-2942

Cat.No: T31553

Synonym: DN1417,DN-1417

Cat.No: T77258

TA 0910 acid-type

Cat.No: T16972

Target: Others

TRH Precursor Peptide

Cat.No: TP2201

Target: Others

Cat.No: T76494

TSHR antagonist S37a

Cat.No: T13217

Target: Others

Prepro-TRH-(160-169)

Cat.No: T76496

TSHR antagonist S37b

Cat.No: T38226

Cat.No: T33438

Synonym: MK-771,MK 771

Cat.No: T70365

Cat.No: T7590

Synonym: TA-0910,他替瑞林

Target: Thyroid hormone receptor(THR)

Cat.No: TP2011

Synonym: JKC 363

Cat.No: T76493

L-Thyroxine-13C9,15N

Cat.No: T36383

Synonym: L-Thyroxine-13C9,15N

Taltirelin-13C-d3

Cat.No: TMIH-0550

Cat. No.	Product Name	Target	Signaling Pathways
T6956	Protirelin Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF	Thyroid hormone receptor(THR); Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Protirelin (Thyroliberin) 是高度保守的神经肽，具有促甲状腺激素水平的激素控制作用，及神经调节功能。

天然产物

Cat.No: T6956

Synonym: Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF

Target: Thyroid hormone receptor(THR), Endogenous Metabolite

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