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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T0128L Vigabatrin Hydrochloride

盐酸氨己烯酸,γ-Vinyl-GABA hydrochloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) 是抑制性神经递质 GABA 乙烯基衍生物,不可逆地抑制 GABA 转氨酶对 GABA 的分解代谢,增加脑中 GABA 的水平。
T64377 AGI-41998 tautomers

Others Others
AGI-41998 tautomers 是pyrido[4,3-d]pyrimidin-7(6H)-one, 8-(4-bromophenyl)-6-(4-methoxyphenyl)-2-[(2,2,2-trifluoroethyl)amino]-. pyrido[4,3-d]pyrimidin-7(6H)-one 的互变异构体。pyrido[4,3-d]pyrimidin-7(6H)-one, 8-(4-bromophenyl)-6-(4-methoxyphenyl)-2-[(2,2,2-trifluoroethyl)amino]-. pyrido[4,3-d]pyrimidin-7(6H)-one 是S-adenosylmethionine synthase isoform type-2抑制剂, IC50= 0.022μM。
T11035 diABZI STING agonist-1 (Tautomerism)

diABZI STING agonist (Compound 3)

STING Immunology/Inflammation
diABZI STING agonist-1 (Tautomerism) (diABZI STING agonist (Compound 3)) 是一个选择性的干扰素基因刺激受体 (STING) 的激动剂,其在人和小鼠中的 EC50 值分别为 130 nM 和 186 nM。。
T13095 Tautomycin

Others Others
Tautomycin is a potent and specific protein phosphatases 1 and 2A inhibitor (Kiapp of 0.16 nM and 0.4 nM for PP1 and PP2A, respectively), and is an antifungal antibiotic isolated from the bacterium Streptomyces verticillatus.

化合物

Vigabatrin Hydrochloride
Cat.No: T0128L
Synonym: 盐酸氨己烯酸,γ-Vinyl-GABA hydrochloride
Target: GABA Receptor
AGI-41998 tautomers
Cat.No: T64377
Synonym:
Target: Others
diABZI STING agonist-1 (Tautomerism)
Cat.No: T11035
Synonym: diABZI STING agonist (Compound 3)
Target: STING
Tautomycin
Cat.No: T13095
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T23421 Tautomycetin

Others Others
protein phosphatase (PP)1 inhibitor

天然产物

Tautomycetin
Cat.No: T23421
Synonym:
Target: Others
TargetMol Loading
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