首页 工具
登录
购物车

搜索结果

Search Results for " tacrolimus monohydrate "
TargetMol的所有产品仅用作科学研究或药证申报,不能被用于人体,我们不向个人提供产品和服务。请您遵守承诺用途,不得违反法律法规规定用于任何其他用途。

3

抑制剂 & 化合物

2

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T71046 FK-1052

FK-1052 is a serotonin 3 & 4 dual receptor antagonist.
T38692 Fabesetron

法贝司琼,FK1052 free base

Fabesetron (FK1052) is an orally active compound that acts as a dual antagonist, targeting both the 5-HT3 and 5-HT4 receptors. It exhibits efficacy in studying emesis induced by cancer chemotherapy, showing potential for managing both acute and delayed symptoms.
T71045 FK-1052 HCl

FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.

化合物

FK-1052
Cat.No: T71046
Synonym:
Target:
Fabesetron
Cat.No: T38692
Synonym: 法贝司琼,FK1052 free base
Target:
FK-1052 HCl
Cat.No: T71045
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T20879 Tacrolimus monohydrate

FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506

Phosphatase; Others; Antibacterial; Antibiotic; Autophagy Autophagy; Metabolism; Microbiology/Virology; Others
Tacrolimus monohydrate (LCP-Tacro) 是大环内酯类化合物,它与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶,从而抑制 T 淋巴细胞信号转导和 IL-2 转录。具有强免疫抑制特性。
T2144 Tacrolimus

他克莫司,Fujimycin,FK506,FR900506

Phosphatase; Others; Antibacterial; Antibiotic; mTOR; Autophagy Autophagy; Metabolism; Microbiology/Virology; Others; PI3K/Akt/mTOR signaling
Tacrolimus (Fujimycin) 可与 FKBP12 结合形成高亲和力复合物 (Ki: 0.2 nM),抑制钙/钙调蛋白依赖性蛋白磷酸酶的活性。

天然产物

Tacrolimus monohydrate
Cat.No: T20879
Synonym: FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506
Target: Phosphatase, Others, Antibacterial, Antibiotic, Autophagy
Tacrolimus
Cat.No: T2144
Synonym: 他克莫司,Fujimycin,FK506,FR900506
Target: Phosphatase, Others, Antibacterial, Antibiotic, mTOR, Autophagy
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼