Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3166 |
VX-11e
Vertex-11e,VTX-11e,TCS ERK 11e |
ERK; GSK-3; FLT; CDK; Aurora Kinase | Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; MAPK; PI3K/Akt/mTOR signaling; Stem Cells; Tyrosine Kinase/Adaptors |
VX-11e (TCS ERK 11e) 是可口服的ERK 高效选择性抑制剂,Ki 值小于 2 nM。 |