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Cat. No. Product Name Target Signaling Pathways
T8866 GW779439X

Apoptosis; Antibacterial; CDK; Aurora Kinase Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Microbiology/Virology
GW779439X 属于吡唑并吡啶类,是一种金黄色葡萄球菌 PASTA 激酶 Stk1抑制剂。它是一种AURKA 抑制剂,可通过 caspases 3/7 诱导细胞凋亡。
T16944 STK16-IN-1

Others Others
STK16-IN-1是一种STK16激酶抑制剂(IC50:295 nM)。
T60946 SLK/STK10-IN-1

SLK/STK10-IN-1 是具有纳摩尔效力的 SLK 和 STK10选择性抑制剂。
T69551 SGC-STK17B-1

SGC-STK17B-1 is a potent and selective inhibitor of STK17B/DRAK2 kinase.
T9473 4SC-203

FLT Angiogenesis; Tyrosine Kinase/Adaptors
4SC-203 是一种具有潜在的抗肿瘤活性的多激酶抑制剂。它对 FLT3/STK1、 FLT3 的突变形式以及 VEGFRs 具有选择性抑制作用。
T71400 Quizartinib HCl

Quizartinib, also know as AC220 and AC010220, is an orally available FLT3 / STK1 inhibitor with potential antineoplastic activity. Class III receptor tyrosine kinase inhibitor AC220 selectively inhibits class III receptor tyrosine kinases, including FMS-related tyrosine kinase 3 (FLT3/STK1), colony-stimulating factor 1 receptor (CSF1R/FMS), stem cell factor receptor (SCFR/KIT), and platelet derived growth factor receptors (PDGFRs), resulting in inhibition of ligand-independent leukemic cell pro...

化合物

GW779439X
Cat.No: T8866
Synonym:
Target: Apoptosis, Antibacterial, CDK, Aurora Kinase
STK16-IN-1
Cat.No: T16944
Synonym:
Target: Others
SLK/STK10-IN-1
Cat.No: T60946
Synonym:
Target:
SGC-STK17B-1
Cat.No: T69551
Synonym:
Target:
4SC-203
Cat.No: T9473
Synonym:
Target: FLT
Quizartinib HCl
Cat.No: T71400
Synonym:
Target:
TargetMol Loading
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