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Cat. No.	Product Name	Target	Signaling Pathways
T0242	Sitagliptin 西他列汀,MK0431,西格列汀	Proteasome; DPP-4; Autophagy	Autophagy; Proteases/Proteasome; Ubiquitination
	Sitagliptin (MK0431) 是一种有效的 DPP4抑制剂，在 Caco-2 细胞中，IC50值为 19 nM。它是一种新型口服降糖药，可单独使用或与二甲双胍或噻唑烷二酮联合用于治疗 2 型糖尿病。
T23358	Sitagliptin phosphate 磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)	DPP-4; Autophagy	Autophagy; Proteases/Proteasome
	Sitagliptin phosphate (MK-0431 phosphate) 是一种二肽基肽酶 4 (DPP4) 抑制剂，在 Caco-2 细胞中，IC50值为 19 nM。
T5903	Sitagliptin Intermediate 2
	Sitagliptin Intermediate 2 是有一种有用的有机化合物，已被用于生命科学相关研究。
T0242L	Sitagliptin phosphate monohydrate MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物	Proteasome; DPP-4; Autophagy	Autophagy; Proteases/Proteasome; Ubiquitination
	Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) 是一种有效的 DPP-IV 抑制剂，在 Caco-2 细胞提取物中的 IC50 为 19 nM。
T40930	(S)-Sitagliptin phosphate (S)-Sitagliptin phosphate,(S)-MK-0431 phosphate
	(S)-Sitagliptin phosphate, the less active S-enantiomer of Sitagliptin phosphate, is a high-potency inhibitor of DPP4. It exhibits an IC50 of 19 nM in Caco-2 cell extracts.
T35440	(-)-Sitagliptin Carbamoyl Glucuronide
	(-)-Sitagliptin carbamoyl glucuronide is a minor phase II metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor (-)-sitagliptin . (-)-Sitagliptin carbamoyl glucuronide is formed by N-carbamoyl glucuronidation and has been found in rat and dog plasma following administration of (-)-sitagliptin.
T35637	Sitagliptin N-Sulfate (sodium salt)
	Sitagliptin N-sulfate is a phase II metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor (-)-sitagliptin . Sitagliptin N-sulfate is formed via sulfation and has been found in rat bile following oral administration of (-)-sitagliptin.
T20028	Janumet Efficib,Janumet XR,Metformin / sitagliptin,Metformin hydrochloride mixture with sitagliptin phosphate
	Metformin hydrochloride mixture with sitagliptin phosphate is an AMP-activated protein kinase stimulant. It is also a CD26 antigen inhibitor, Gluconeogenesis inhibitor, and Glucose modulator.
T63915	Sitagliptin fenilalanil
	Sitagliptin fenilalanil 是一种二肽氨基肽酶 (DPP-4)抑制剂。
T74592	Sitagliptin fenilalanil hydrochloride
	Sitagliptin fenilalanil hydrochloride 是一种二肽氨基肽酶 (DPP-4) 抑制剂。
T63166L	(S, R)-LSN 3318839 (S, R)-LSN 3318839(Isomer-2764704-18-7)	Glucagon Receptor	GPCR/G Protein

T70373	AS2575959
	AS2575959 is a novel GPR40 agonist, exhibiting glucose metabolism improvement and synergistic effect with sitagliptin on insulin and incretin secretion.
T37522	Teneligliptin
	Teneligliptin (MP-513) is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM. Teneligliptin (MP-513) inhibits all these DPP-4 enzymes in a concentration-dependent manner. The IC50s of Teneligliptin (MP-513) for rhDPP-4, human plasma, and rat plasma are 0.889, 1.75, and 1.35 nM, respectively. A study of enzyme inhibition kinetics is conducted for Teneligliptin (M...

化合物

Cat.No: T0242

Synonym: 西他列汀,MK0431,西格列汀

Target: Proteasome, DPP-4, Autophagy

Sitagliptin phosphate

Cat.No: T23358

Synonym: 磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)

Target: DPP-4, Autophagy

Sitagliptin Intermediate 2

Cat.No: T5903

Sitagliptin phosphate monohydrate

Cat.No: T0242L

Synonym: MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物

Target: Proteasome, DPP-4, Autophagy

(S)-Sitagliptin phosphate

Cat.No: T40930

Synonym: (S)-Sitagliptin phosphate,(S)-MK-0431 phosphate

(-)-Sitagliptin Carbamoyl Glucuronide

Cat.No: T35440

Sitagliptin N-Sulfate (sodium salt)

Cat.No: T35637

Cat.No: T20028

Synonym: Efficib,Janumet XR,Metformin / sitagliptin,Metformin hydrochloride mixture with sitagliptin phosphate

Sitagliptin fenilalanil

Cat.No: T63915

Sitagliptin fenilalanil hydrochloride

Cat.No: T74592

(S, R)-LSN 3318839

Cat.No: T63166L

Synonym: (S, R)-LSN 3318839(Isomer-2764704-18-7)

Target: Glucagon Receptor

Cat.No: T70373

Cat.No: T37522

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