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Cat. No. Product Name Target Signaling Pathways
T12908 SIBA

5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine,5ˊ-异丁硫基-5ˊ-脱氧腺苷

Nucleoside Antimetabolite/Analog; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
SIBA (5'-Deoxy-5'-isobutylthioadenosine) 是 SAH 的合成类似物,可作为 S-腺苷甲硫氨酸介导的甲基转移的抑制剂。它干扰多种酶活性,可逆地阻断单纯疱疹病毒 1 型病毒的繁殖。
T4996 Atosiban

阿托西班,RWJ22164,RW22164

Oxytocin Receptor; Vasopressin Receptor Endocrinology/Hormones; GPCR/G Protein
Atosiban (RW22164) 是一种脱氨基催产素类似物,是一种九肽,也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂,可用于自发早产的研究。
T5148 Atosiban acetate

RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班

Oxytocin Receptor; Vasopressin Receptor Endocrinology/Hormones; GPCR/G Protein
Atosiban acetate (RW22164) 是一种脱氨基催产素类似物,是一种九肽,也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂,可用于自发早产的研究。
T70570 Erlosiban

Erlosiban, also known as OBE001, is a novel, orally active nonpeptide oxytocin receptor antagonist under development for the treatment of preterm labor and improvement in embryo implantation and pregnancy rate in assisted reproductive technology (ART).
T16736 Retosiban

GSK 221149,GSK 221149A

Others Others
Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).
T69504 Barusiban

Barusiban is an oxytocin receptor antagonist.
T11502 Epelsiban

GSK 557296

Others Others
Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).
T31647 Epelsiban besylate

GSK-557296B,GSK557296B

Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.

化合物

SIBA
Cat.No: T12908
Synonym: 5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine,5ˊ-异丁硫基-5ˊ-脱氧腺苷
Target: Nucleoside Antimetabolite/Analog, HSV
Atosiban
Cat.No: T4996
Synonym: 阿托西班,RWJ22164,RW22164
Target: Oxytocin Receptor, Vasopressin Receptor
Atosiban acetate
Cat.No: T5148
Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班
Target: Oxytocin Receptor, Vasopressin Receptor
Erlosiban
Cat.No: T70570
Synonym:
Target:
Retosiban
Cat.No: T16736
Synonym: GSK 221149,GSK 221149A
Target: Others
Barusiban
Cat.No: T69504
Synonym:
Target:
Epelsiban
Cat.No: T11502
Synonym: GSK 557296
Target: Others
Epelsiban besylate
Cat.No: T31647
Synonym: GSK-557296B,GSK557296B
Target:
TargetMol Loading
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