Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T40207 | SARS-CoV-2-IN-7 | ||
SARS-CoV-2-IN-7 demonstrates potent inhibition of viral replication in SARS-CoV-2-infected Vero E6 cells with an IC50 value of 844 nM. | |||
T79278 |
SARS-CoV-2 Mpro-IN-7
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SARS-CoV | Microbiology/Virology |
Mpro-IN-7(化合物6g)是一种针对Mpro-SARS-CoV-2的高效抑制剂,具有IC50值为8.8 μM,CC50值为10 μM。 | |||
T72371 |
SARS-CoV-2 3CLpro-IN-7
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SARS-CoV-2 3CLpro-IN-7 是一种可逆的共价SARS-CoV-2 3CL 蛋白酶抑制剂,IC50值为 1.4 µM。 | |||
T9287 |
Hydroxychloroquine
2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol,羟氯喹 |
SARS-CoV; TLR; Parasite; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology |
Hydroxychloroquine (2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol) 是一种合成抗疟疾剂,有效抑制SARS-CoV-2感染,也抑制 Toll 样受体 7/9 信号传导。 | |||
T0951 |
Hydroxychloroquine sulfate
Acidum iopanoicum,硫酸羟基氯喹,硫酸羟氯喹,HCQ sulfate |
DNA; SARS-CoV; TLR; Parasite; Autophagy | Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology |
Hydroxychloroquine sulfate (Acidum iopanoicum) 抑制疟原虫血红素聚合酶。它还可抑制 Toll 样受体 7/9 信号传导和 SARS-CoV-2 感染。 | |||
T78725 | SARS-CoV-2 nsp14-IN-3 | SARS-CoV | Microbiology/Virology |
SARS-CoV-2 nsp14-IN-3 (4975)为一种针对SARS-CoV-2 Nsp14 N7-甲基转移酶的抑制剂,具有IC50值为7 μM。 | |||
T69536 |
MMT5-14
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MMT5-14 is a SARS-CoV-2 inhibitor. MMT5-14 showed 2- to 7-fold higher antiviral activity in four variants of SARS-CoV-2. By reducing premature hydrolysis in hamsters, MMT5-14 increased the prodrug concentration by 200- to 300-fold in the plasma and lungs but also enhanced lung accumulation of the active metabolite triphosphate nucleosides (NTP) by 5-fold. | |||
T73964 | Hydroxychloroquine Impurity F | ||
Hydroxychloroquine Impurity F为Hydroxychloroquine的一种杂质,后者为合成抗疟疾剂,能抑制Toll样受体7/9(TLR7/9)信号传导,并有效抑制SARS-CoV-2感染。 | |||
T73963 |
Hydroxychloroquine Impurity E
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Hydroxychloroquine Impurity E, Hydroxychloroquine的一种杂质,属于合成抗疟疾剂,能抑制Toll样受体7/9 (TLR7/9) 信号传递,且对抗SARS-CoV-2感染有效。 | |||
T79234 |
RdRP-IN-7
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SARS-CoV | Microbiology/Virology |
RdRP-IN-7是一种抑制剂,针对RNA依赖性RNA聚合酶(RdRP),对SARS-CoV-2有抑制效果,IC50为8.2μM,IC90为14.1μM,并且CC90为79.1μM。该化合物适用于抗病毒研究。 | |||
T38174 | Mpro inhibitor N3 hemihydrate | ||
Mpro inhibitor N3 hemihydrate is a potent inhibitor of SARS-CoV-2 Mpro with an EC50 of 16.77 μM for SARS-CoV-2. Mpro inhibitor N3 hemihydrate specifically inhibits Mpro from multiple coronaviruses, including SARS-CoV and MERS-CoV. Mpro inhibitor N3 hemihydrate displays inhibition against HCoV-229E, FIPV, and MHV-A59 with individual IC50 of 4.0 μM, 8.8 μM, and 2.7 μM, respectively[1][2]. Mpro inhibitor N3 hemihydrate (0-0.64 μM) is able to penetrate cells to inhibit the replication of IBV viruses... | |||
TMIH-0146 |
Chloroquine-d5
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Chloroquine-d5 是 Chloroquine 的氘代化合物。Chloroquine 的 CAS 号为 54-05-7。Chloroquine 是一种自噬和 Toll 样受体抑制剂。 氯喹是一种抗疟疾和抗炎剂,广泛用于治疗疟疾和类风湿性关节炎。它在体外控制 SARS-CoV-2 (COVID-19) 感染方面非常有效,EC50 为 1.13 μM。 |