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Cat. No. Product Name Target Signaling Pathways
T6955 Propafenone hydrochloride

Propafenone HCl,Arythmol,SA-79 (hydrochloride),Rytmonorm,盐酸普罗帕酮,Rythmol

Sodium Channel Membrane transporter/Ion channel
Propafenone hydrochloride (Arythmol8) 具有抗心律不齐的功效,可用于心房和心室性心律不齐。
T0866 Propafenone

Rythmol,普罗帕酮,Propafenonum

Potassium Channel; MRP; Sodium Channel Immunology/Inflammation; Membrane transporter/Ion channel
Propafenone (Propafenonum) 是钠通道阻滞剂,它对 β 受体具有高亲和力 (IC50=32 nM)。它能够阻断瞬时外向钾电流 (Ito) (IC50: 4.9 nM) 和持续延迟整流器K+电流 (Isus) (IC50: 8.6 nM) ,具有抗心律失常的作用。它能够诱导线粒体功能障碍及诱导细胞凋亡,从而抑制食管癌增殖。
T12811 (S)-Propafenone

(S)-SA-79

Others Others
(S)-Propafenone ((S)-SA-79) is the S-enantiomer of Propafenone. It possesses beta-blocking properties and exhibits class 1 antiarrhythmic activity reliant on sodium channel blockade.
T12548 Propafenone D7 hydrochloride

盐酸普罗帕酮 D7,SA-79 (D7 hydrochloride)

Others Others
Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.

化合物

Propafenone hydrochloride
Cat.No: T6955
Synonym: Propafenone HCl,Arythmol,SA-79 (hydrochloride),Rytmonorm,盐酸普罗帕酮,Rythmol
Target: Sodium Channel
Propafenone
Cat.No: T0866
Synonym: Rythmol,普罗帕酮,Propafenonum
Target: Potassium Channel, MRP, Sodium Channel
(S)-Propafenone
Cat.No: T12811
Synonym: (S)-SA-79
Target: Others
Propafenone D7 hydrochloride
Cat.No: T12548
Synonym: 盐酸普罗帕酮 D7,SA-79 (D7 hydrochloride)
Target: Others
TargetMol Loading
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