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Cat. No. Product Name Target Signaling Pathways
T6252 Ipatasertib

GDC-0068,RG7440,帕他色替

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Ipatasertib (GDC-0068) 是选择性的,ATP 竞争性的pan-Akt 抑制剂,能够抑制Akt1 (IC50:5 nM),Akt2 (IC50:18 nM),Akt3 (IC50:8 nM)。
T18053 Ipatasertib-NH2

RG7440-NH2,GDC-0068-NH2

Others Others
Ipatasertib-NH2 (GDC-0068-NH2;RG7440-NH2) is a ligand for target protein AKT for PROTAC, binds to lenalidomide, a ligand of ubiquitin E3 ligase cereblon (CRBN), via a ten-hydrocarbon linker to form INY-03-041 to degrade AKT[1].
T38393 Ipatasertib-NH2 dihydrochloride

RG7440-NH2 dihydrochloride,Ipatasertib-NH2 dihydrochloride,GDC-0068-NH2 dihydrochloride

Ipatasertib-NH2 dihydrochloride is a ligand for the target protein AKT in PROTAC INY-03-041. INY-03-041 consists of Ipatasertib-NH2, a ten-hydrocarbon linker, and the CRBN ligand Lenalidomide, which acts as an E3 ubiquitin ligase.
T27621 Ipatasertib HCl

GDC0068,RG 7440,GDC 0068,RG-7440,GDC-0068,RG7440

Ipatasertib is an orally active, potent and selective Akt inhibitor with antitumor activity. Inhibition of Akt activity by Ipatasertib resulted in blockade of cell-cycle progression and reduced viability of cancer cell lines. Markers of Akt activation, in
T15374 Ipatasertib dihydrochloride

GDC-0068 dihydrochloride,RG-7440 dihydrochloride

Akt; PKA Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) 是ATP 竞争性的pan-Akt 选择性抑制剂,抑制Akt1,Akt2,Akt3,IC50分别为 5,18,8 nM。
T70550 BMS-986034

BMS-986034 is a GPR119 agonist.

化合物

Ipatasertib
Cat.No: T6252
Synonym: GDC-0068,RG7440,帕他色替
Target: Akt
Ipatasertib-NH2
Cat.No: T18053
Synonym: RG7440-NH2,GDC-0068-NH2
Target: Others
Ipatasertib-NH2 dihydrochloride
Cat.No: T38393
Synonym: RG7440-NH2 dihydrochloride,Ipatasertib-NH2 dihydrochloride,GDC-0068-NH2 dihydrochloride
Target:
Ipatasertib HCl
Cat.No: T27621
Synonym: GDC0068,RG 7440,GDC 0068,RG-7440,GDC-0068,RG7440
Target:
Ipatasertib dihydrochloride
Cat.No: T15374
Synonym: GDC-0068 dihydrochloride,RG-7440 dihydrochloride
Target: Akt, PKA
BMS-986034
Cat.No: T70550
Synonym:
Target:
TargetMol Loading
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