Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2116 |
Pteropodine
|
BCL; Calcium Channel; 5-HT Receptor | Apoptosis; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Pteropodine acts as a positive modulator of muscarinic M(1) and 5-HT(2) receptors. Pteropodine shows antigenotoxic, antioxidant and lymphocyte induction effects, it also shows strong apoptotic effect on acute leukaemic lymphoblasts. | |||
TN1790 |
Isopteropodine
Uncarine E |
5-HT Receptor; Antibacterial; AChR | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Isopteropodine (Uncarine E) 是从 Hamelia patens micropropagated 分离得到的一种异育亨宾型辛吲哚生物碱.具有抗菌活性,可刺激机体免疫系统。Isopteropodine 是 M1 型毒蕈碱乙酰胆碱 (muscarinic M1) 受体及 5-HT2 受体的正向调节剂,是PXR激活剂,可诱导大鼠子宫肌层收缩。 | |||
TN4311 |
Isomitraphylline
|
Others | Others |
Isomitraphylline and pteropodine are the most suitable for standardization of medical cat's claw preparations. Isomitraphylline can inhibit proliferation of acute lymphoblastic leukaemia cells. |