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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3695 Pepstatin

抑肽素,Pepstatin A,Pepsin Inhibitor S 735A,Ahpatinin C

Amino Acids and Derivatives; Proteasome; HIV Protease; Autophagy Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome; Ubiquitination
Pepstatin (Pepsin Inhibitor S 735A) 是由放线菌类产生的特异性天冬氨酸蛋白酶抑制剂,可抑制 HIV 蛋白酶的活性。
T12407 Pepstatin Ammonium

Pepstatin A Ammonium

Others Others
Pepstatin Ammonium is a specific inhibitor of aspartic proteaseproduced by actinomycetes(hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease with IC50s of 4.5 nM, 6.2 nM, 150 nM, 290 nM
T26302 Tyrostatin

N-Isovaleryl-tyrosyl-leucyl-tyrosinal

Tyrostatin is a new pepstatin-insensitive carboxyl proteinases peptide proteinase inhibitor isolated from Kitasatosporia.
T25938 Pepstanone A

Pepstanone A is a potent aspartyl protease inhibitor, produced by pepstatin-producing Streptomyces.

化合物

Pepstatin
Cat.No: T3695
Synonym: 抑肽素,Pepstatin A,Pepsin Inhibitor S 735A,Ahpatinin C
Target: Amino Acids and Derivatives, Proteasome, HIV Protease, Autophagy
Pepstatin Ammonium
Cat.No: T12407
Synonym: Pepstatin A Ammonium
Target: Others
Tyrostatin
Cat.No: T26302
Synonym: N-Isovaleryl-tyrosyl-leucyl-tyrosinal
Target:
Pepstanone A
Cat.No: T25938
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T75705 Pepstatin Trifluoroacetate

Pepstatin (Pepstatin A) Trifluoroacetate 是一种由放线菌产生的特异性天冬氨酸蛋白酶(aspartic proteases)抑制剂,口服活性强。该化合物能有效抑制hemoglobin-pepsin、hemoglobin-proctase、casein-pepsin、casein-proctase、casein-acid protease和hemoglobin-acid protease的活性,其IC50值分别为4.5 nM、6.2 nM、150 nM、290 nM、520 nM和260 nM。此外,对HIV protease也有抑制作用。

天然产物

Pepstatin Trifluoroacetate
Cat.No: T75705
Synonym:
Target:
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