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Cat. No. Product Name Target Signaling Pathways
T23133 Pentamidine

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine 是抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T1654 Pentamidine isethionate

Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine isethionate (Pentamidine diisethionate) 是抗微生物剂,会干扰 DNA 的生物合成。它抑制寄生虫Leishmania infantum,IC50为 2.5 μM。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它有抗肿瘤和抗菌活性。
T23132 Pentamidine dihydrochloride

喷他脒二盐酸盐,MP-601205 dihydrochloride

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine dihydrochloride (MP-601205 dihydrochloride) 是一种抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T28355 Pentamidine dimesylate

Pentamidine dimesylate is an inhibitor of calcium-dependent complex formation with p53 [(Ca)S100B-p53) in malignant melanoma (MM). Pentamidine dimesylate restores p53 tumor suppressor activity in vivo.
T11553 Heptamidine dimethanesulfonate

SBi4211 dimethanesulfonate

Others Others
Heptamidine dimethanesulfonate (SBi4211 dimethanesulfonate) 是一种与喷他脒有关的、强效的钙结合蛋白 S100B 的抑制剂 (Kd=6.9 μM),选择性地杀死表达 S100B 的黑素瘤细胞。它是有效的强直性肌营养不良 (DM) 研究工具。
T11553L Heptamidine

SBi4211

Others Others
Heptamidine is an effective Pentamidine-related inhibitor of the calcium-binding protein S100B (Kd: 6.9 μM). It selectively kills melanoma cells with S100B over those without S100B. It is a useful tool for the investigation of Myotonic dystrophy.

化合物

Pentamidine
Cat.No: T23133
Synonym:
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Pentamidine isethionate
Cat.No: T1654
Synonym: Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Pentamidine dihydrochloride
Cat.No: T23132
Synonym: 喷他脒二盐酸盐,MP-601205 dihydrochloride
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Pentamidine dimesylate
Cat.No: T28355
Synonym:
Target:
Heptamidine dimethanesulfonate
Cat.No: T11553
Synonym: SBi4211 dimethanesulfonate
Target: Others
Heptamidine
Cat.No: T11553L
Synonym: SBi4211
Target: Others
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