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Cat. No. Product Name Target Signaling Pathways
T39901 PROTAC IRAK4 degrader-4

PROTAC IRAK4 degrader-4

PROTAC IRAK4 degrader-4 (US20190192668A1, compound I-127) is a Cereblon-based PROTAC specifically designed to target and degrade interleukin-1 receptor-associated kinase 4 (IRAK4).
T39902 PROTAC IRAK4 degrader-5

PROTAC IRAK4 degrader-5

PROTAC IRAK4 degrader-5 is a Cereblon-based IRAK4 degrader.
T39903 PROTAC IRAK4 degrader-6

PROTAC IRAK4 degrader-6

PROTAC IRAK4 degrader-6 is a potent Cereblon-based compound designed to degrade interleukin-1 receptor-associated kinase 4 (IRAK4).
T39920 PROTAC IRAK4 degrader-3

PROTAC IRAK4 degrader-3

PROTACs PROTAC
PROTAC IRAK4 degrader-3 is a PROTAC-induced IRAK4 degrader based on von Hippel-Lindau.
T13842 PROTAC IRAK4 degrader-1

Others; PROTACs Others; PROTAC
PROTAC IRAK4 degrader-1 is a degrader of PROTAC interleukin-1 receptor-associated kinase 4 (IRAK4).
T7755 Thalidomide 4-fluoride

E3 ligase Ligand 4,2-(2,6-二氧代-哌啶-3-基)-4-氟基-异吲哚-1,3-二酮

IRAK; Ligand for E3 Ligase Immunology/Inflammation; NF-κB; PROTAC
Thalidomide 4-fluoride (E3 ligase Ligand 4) 是一种基于 Thalidomide 的 Cereblon 配体,可用于募集 CRBN 蛋白。它能够利用 linker 与 IRAK4 靶蛋白配体连接,得到 PROTAC IRAK4 degrader-1。

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PROTAC IRAK4 degrader-4
Cat.No: T39901
Synonym: PROTAC IRAK4 degrader-4
Target:
PROTAC IRAK4 degrader-5
Cat.No: T39902
Synonym: PROTAC IRAK4 degrader-5
Target:
PROTAC IRAK4 degrader-6
Cat.No: T39903
Synonym: PROTAC IRAK4 degrader-6
Target:
PROTAC IRAK4 degrader-3
Cat.No: T39920
Synonym: PROTAC IRAK4 degrader-3
Target: PROTACs
PROTAC IRAK4 degrader-1
Cat.No: T13842
Synonym:
Target: Others, PROTACs
Thalidomide 4-fluoride
Cat.No: T7755
Synonym: E3 ligase Ligand 4,2-(2,6-二氧代-哌啶-3-基)-4-氟基-异吲哚-1,3-二酮
Target: IRAK, Ligand for E3 Ligase
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