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Cat. No. Product Name Target Signaling Pathways
T1264 Ciprofibrate

Win35833,环丙贝特

PPAR DNA Damage/DNA Repair; Metabolism
Ciprofibrate (Win35833) 是一种有效的过氧化物酶体增殖物,可增加PPARα的磷酸化水平。它是一种可口服的降血脂剂,可研究原发性高脂血症。
T70289 Terpendole E

Terpendole E is an atypical L5 site inhibitor.
T10900 CUDA

PPAR; Epoxide Hydrolase DNA Damage/DNA Repair; Metabolism
CUDA 是一种可溶性环氧水解酶抑制剂,对小鼠 sEH 和人 sEH 作用的 IC50分别为 11.1 和 112 nM。它能选择性地上调过氧化物酶体增殖激活受体 PPARα的活性,有用于心血管疾病的研究潜力。
T10505 PPARα-MO-1

PPAR DNA Damage/DNA Repair; Metabolism
PPARα-MO-1 is a potent modulator of PPARα.
T1415 Gemfibrozil

吉非罗齐,CI-719,Jezil,Decrelip,Lopid

P450; Adrenergic Receptor; PPAR DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience
Gemfibrozil (CI-719) 是一种PPAR-α激活剂,可作为降脂药。它也是P450非选择性抑制剂,对 CYP2C9、2C19、2C8 和 1A2 的Ki 值分别为 5.8、24、69 和 82 μM。
T5532 BMS-687453

PPAR DNA Damage/DNA Repair; Metabolism
BMS-687453 是一种选择性 PPARα激动剂,对人 PPARα的 EC50和 IC50分别为 10 nM 和 260 nM。它较弱地抑制 PPARγ 的活性,EC50和 IC50值分别为 4100 nM 和大于 15000 nM。
T25198 C-333H

C333H

C-333H is a new PPARalpha/gamma dual agonist.
T70141 MDK80908

MDK80908, also known as PPARalpha/gamma agonist N15, is a dual PPARα/γ agonist, ameliorating insulin resistance and gluconeogenesis in vivo and vitro. MDK80908 has CAS#1821380-90-8.
T70290 YUN90389

YUN90389, also known as PPARalpha/delta-IN-11, is a the first reported pparα/δ dual antagonist. YUN90389 was first reported in Bioorganic & Medicinal Chemistry Letters (2019), 29(3), 503-508. YUN90389 has CAS#1673590-38-9. This product has no formal name at the moment. For the convenience of communication, a temporary code name was therefore proposed according to MedKoo Chemical Nomenclature (see web page: https://www.medkoo.com/page/naming).

化合物

Ciprofibrate
Cat.No: T1264
Synonym: Win35833,环丙贝特
Target: PPAR
Terpendole E
Cat.No: T70289
Synonym:
Target:
CUDA
Cat.No: T10900
Synonym:
Target: PPAR, Epoxide Hydrolase
PPARα-MO-1
Cat.No: T10505
Synonym:
Target: PPAR
Gemfibrozil
Cat.No: T1415
Synonym: 吉非罗齐,CI-719,Jezil,Decrelip,Lopid
Target: P450, Adrenergic Receptor, PPAR
BMS-687453
Cat.No: T5532
Synonym:
Target: PPAR
C-333H
Cat.No: T25198
Synonym: C333H
Target:
MDK80908
Cat.No: T70141
Synonym:
Target:
YUN90389
Cat.No: T70290
Synonym:
Target:
TargetMol Loading
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