Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1264 |
Ciprofibrate
Win35833,环丙贝特 |
PPAR | DNA Damage/DNA Repair; Metabolism |
Ciprofibrate (Win35833) 是一种有效的过氧化物酶体增殖物,可增加PPARα的磷酸化水平。它是一种可口服的降血脂剂,可研究原发性高脂血症。 | |||
T70289 |
Terpendole E
|
||
Terpendole E is an atypical L5 site inhibitor. | |||
T10900 |
CUDA
|
PPAR; Epoxide Hydrolase | DNA Damage/DNA Repair; Metabolism |
CUDA 是一种可溶性环氧水解酶抑制剂,对小鼠 sEH 和人 sEH 作用的 IC50分别为 11.1 和 112 nM。它能选择性地上调过氧化物酶体增殖激活受体 PPARα的活性,有用于心血管疾病的研究潜力。 | |||
T10505 | PPARα-MO-1 | PPAR | DNA Damage/DNA Repair; Metabolism |
PPARα-MO-1 is a potent modulator of PPARα. | |||
T1415 |
Gemfibrozil
吉非罗齐,CI-719,Jezil,Decrelip,Lopid |
P450; Adrenergic Receptor; PPAR | DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience |
Gemfibrozil (CI-719) 是一种PPAR-α激活剂,可作为降脂药。它也是P450非选择性抑制剂,对 CYP2C9、2C19、2C8 和 1A2 的Ki 值分别为 5.8、24、69 和 82 μM。 | |||
T5532 |
BMS-687453
|
PPAR | DNA Damage/DNA Repair; Metabolism |
BMS-687453 是一种选择性 PPARα激动剂,对人 PPARα的 EC50和 IC50分别为 10 nM 和 260 nM。它较弱地抑制 PPARγ 的活性,EC50和 IC50值分别为 4100 nM 和大于 15000 nM。 | |||
T25198 |
C-333H
C333H |
||
C-333H is a new PPARalpha/gamma dual agonist. | |||
T70141 | MDK80908 | ||
MDK80908, also known as PPARalpha/gamma agonist N15, is a dual PPARα/γ agonist, ameliorating insulin resistance and gluconeogenesis in vivo and vitro. MDK80908 has CAS#1821380-90-8. | |||
T70290 | YUN90389 | ||
YUN90389, also known as PPARalpha/delta-IN-11, is a the first reported pparα/δ dual antagonist. YUN90389 was first reported in Bioorganic & Medicinal Chemistry Letters (2019), 29(3), 503-508. YUN90389 has CAS#1673590-38-9. This product has no formal name at the moment. For the convenience of communication, a temporary code name was therefore proposed according to MedKoo Chemical Nomenclature (see web page: https://www.medkoo.com/page/naming). |