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6

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6266 PP2

AGL 1879,AG 1879,AGL 1879

EGFR; Tyrosine Kinases; JAK; Src Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
PP2 (AG 1879,AGL 1879) 是 Lck/Fyn 抑制剂 (IC50:4/5 nM),对 EGFR 的效力降低约 100 倍,对 ZAP-70、PKA 和 JAK2 无活性。
T6266L PP2 Analog

PP2-Analog,CHEMBL-306012,CHEMBL306012,CHEMBL 306012

PP2 Analog is an analog of PP2. It also acts as a protein trafficking modulator.
T70131 TPP2a bromide

TPP2a is a mitochondrial thioredoxin reductase (TrxR) inhibitor.
T63259 PP2A Cancerous-IN-1

PP2A Cancerous-IN-1 是强效的 CIP2A(Cancerous inhibitor of PP2A) 和 p-Akt 抑制剂,表现出强大的抗增殖作用。
T82671 CPP2

CPP2为一种具备高细胞内易位效率的细胞穿透肽。
T77976 PROTAC Her3 Degrader-8

PROTACs PROTAC
PROTACHer3 Degrader-8(Compound PP2)是一类PROTAC,能在体外及细胞实验中降解Her3蛋白,适用于HER家族蛋白调控的疾病研究。

化合物

PP2
Cat.No: T6266
Synonym: AGL 1879,AG 1879,AGL 1879
Target: EGFR, Tyrosine Kinases, JAK, Src
PP2 Analog
Cat.No: T6266L
Synonym: PP2-Analog,CHEMBL-306012,CHEMBL306012,CHEMBL 306012
Target:
TPP2a bromide
Cat.No: T70131
Synonym:
Target:
PP2A Cancerous-IN-1
Cat.No: T63259
Synonym:
Target:
CPP2
Cat.No: T82671
Synonym:
Target:
PROTAC Her3 Degrader-8
Cat.No: T77976
Synonym:
Target: PROTACs
Cat. No. Product Name Target Signaling Pathways
T16381 Okadaic acid

Others Others
Okadaic acid is a non-comepetitive, selective and reversible serine/threonine-specific protein phosphatases 1 (PP1), PP2A, and PP3 inhibitor (IC50s: 10-15 nM, 0.5 nM, and 4 nM, respectively). Okadaic acid is extracted from black sponges of the genus Halic

天然产物

Okadaic acid
Cat.No: T16381
Synonym:
Target: Others
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