Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3440 |
2-PMPA
2-(Phosphonomethyl)pentanedioic acid |
Carboxypeptidase | Proteases/Proteasome |
2-PMPA (2-(Phosphonomethyl)pentanedioic acid) 是谷氨酸羧肽酶II 的选择性抑制剂(IC50:300 pM)。 | |||
T25968 |
PMPA sodium
PMPA sodium salt,PMPA tetrasodium salt,PMPA Na |
||
PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor. | |||
T7111 |
Tenofovir Disoproxil
替诺福韦酯,GS 4331,Bis(POC)-PMPA |
HBV; HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Tenofovir Disoproxil (GS 4331) 是一种核苷酸逆转录酶抑制剂,用于治疗 HIV 和慢性乙型肝炎。 | |||
T12814 |
(S)-Tenofovir
(S)-替诺福韦,(S)-PMPA,(S)-GS 1278,(S)-TDF |
Others | Others |
(S)-Tenofovir ((S)-PMPA) 是Tenofovir 的活性较低的S-对映体,Tenofovir 是一种核苷酸逆转录酶抑制剂。 | |||
T23165 |
PMPA (NMDA antagonist)
|
Others | Others |
PMPA (NMDA antagonist) is a Competitive NMDA receptor antagonist. | |||
T1649 |
Tenofovir
替诺福韦,泰诺福韦,PMPA,TDF,GS 1278 |
HBV; HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Tenofovir (GS 1278) 是一种核苷酸逆转录酶抑制剂,可研究 HIV 和慢性乙型肝炎。 | |||
T2409L |
Tenofovir Disoproxil Fumarate
GS-1278 Disoproxil Fumarate,Tenofovir DF,富马酸替诺福韦酯 |
HBV; HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Tenofovir Disoproxil Fumarate (GS-1278 Disoproxil Fumarate) 是一种核苷酸逆转录酶抑制剂,有潜力研究艾滋病和慢性乙型肝炎。 | |||
T67798 |
(2RS)-FPMPA
FPMPA |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
(2RS)-FPMPA(FPMPA) 具有抗病毒活性,在感染SHIV(DH4R)的人MT12细胞的测得IC50 值为1.85μM。 | |||
T67820 | FPMPA PM | ||
FPMPA PM 是 FPMPA 的衍生物。FPMPA 是一种选择性腺苷 A3受体激动剂,具有抗炎、镇痛和神经保护活性。 | |||
T23467 |
TPMPA
|
Others | Others |
GABAA-ρ antagonist | |||
T14488 |
Azt-pmap
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1]. As a nucleoside reverse transcriptase inhibitor (NRTI), AZT-PMPA targets HIV infection effectively[2]. |