Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6251 |
PF-04691502
PF4691502 |
Akt; PI3K; mTOR; Autophagy | Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
PF-04691502 是一种有效的选择性 PI3K 和 mTOR 激酶抑制剂,具有抗肿瘤活性。它与人 PI3Kα、β、δ、γ和 mTOR 结合的 Ki 分别为1.8、2.1、1.6、1.9和16 nM。 | |||
T28373 |
PF-06465603
PF06465603,PF 06465603 |
||
PF-06465603 is a metabolite of PF-04691502, a highly potent and selective ATP competitive kinase inhibitor of class 1 PI3Ks and mTOR. |