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Cat. No. Product Name Target Signaling Pathways
T1308 Orphenadrine hydrochloride

Mebedrol,Mephenamin,盐酸邻甲苯海拉明

Sodium Channel; NMDAR; Norepinephrine; iGluR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Orphenadrine hydrochloride (Mephenamin) 是一种非竞争性的NMDA 受体拮抗剂, Ki=6.0 ± 0.7 μM。
T71537 Tofenacin hydrochloride

Tofenacin hydrochloride is an antidepressant drug with a tricyclic-like structure. It acts as a serotonin-norepinephrine reuptake inhibitor, and based on its close relation to orphenadrine, may also possess anticholinergic and antihistamine properties. Tofenacin is also the major active metabolite of orphenadrine and likely plays a role in its beneficial effects against depressive symptoms seen in Parkinson's disease patients.

化合物

Orphenadrine hydrochloride
Cat.No: T1308
Synonym: Mebedrol,Mephenamin,盐酸邻甲苯海拉明
Target: Sodium Channel, NMDAR, Norepinephrine, iGluR, Histamine Receptor
Tofenacin hydrochloride
Cat.No: T71537
Synonym:
Target:
TargetMol Loading
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