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Cat. No. Product Name Target Signaling Pathways
T3183 SAX-187

WAY 181187,WAY181187

5-HT Receptor GPCR/G Protein; Neuroscience
SAX-187 (SAX-187) 是一种有效的选择性5-HT6受体激动剂,Ki 为 2.2 nM,EC50为 6.6 nM。它介导 5-HT6 受体依赖性信号通路,可作为特异性激动剂。
T0255 Clomipramine hydrochloride

Clomipramine HCl,Anafranil,盐酸氯米帕明

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine; GST GPCR/G Protein; Neuroscience; oxidation-reduction
Clomipramine hydrochloride (Anafranil) 是一种5-羟色胺转运体(Ki:0.14 nM)、去甲肾上腺素转运体(Ki:54 nM)和多巴胺转运体(Ki:3 nM)阻断剂。
T21013 Clomipramine

Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明

5-HT Receptor GPCR/G Protein; Neuroscience
Clomipramine (Clomicalm) 是一种三环类抗抑郁药,能够有效阻断 5-HT 再摄取 (IC50:1.5 nM) ,可用于研究强迫症 (OCD) 及抑郁症。
T82271 Golocdacimab

MEDI6570

Golocdacimab (MEDI6570) 是一种针对LOX-1的全人源单克隆抗体,潜在可用于研究2型糖尿病。
T68683 Sertraline Free Base

Sertraline Free Base is a Selective Serotonin Reuptake Inhibitor (SSRI). It can treat depression, obsessive-compulsive disorder (OCD), posttraumatic stress disorder (PTSD), premenstrual dysphoric disorder (PMDD), social anxiety disorder, and panic disorder.
T68579 Fluvoxamine acid

Fluvoxamine acid is a medication which functions as a selective serotonin reuptake inhibitor (SSRI) and σ1 receptor agonist. Fluvoxamine is used primarily for the treatment of obsessive-compulsive disorder (OCD), and is also used to treat major depressive disorder (MDD), and anxiety disorders such as panic disorder and post-traumatic stress disorder (PTSD).

化合物

SAX-187
Cat.No: T3183
Synonym: WAY 181187,WAY181187
Target: 5-HT Receptor
Clomipramine hydrochloride
Cat.No: T0255
Synonym: Clomipramine HCl,Anafranil,盐酸氯米帕明
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine, GST
Clomipramine
Cat.No: T21013
Synonym: Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明
Target: 5-HT Receptor
Golocdacimab
Cat.No: T82271
Synonym: MEDI6570
Target:
Sertraline Free Base
Cat.No: T68683
Synonym:
Target:
Fluvoxamine acid
Cat.No: T68579
Synonym:
Target:
TargetMol Loading
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