Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16324 |
Nimbolide
|
Apoptosis; NF-κB; CDK | Apoptosis; Cell Cycle/Checkpoint; NF-κB |
Nimbolide 是源自印楝叶和花的一种三萜。它抑制CDK4/CDK6激酶活性。它抑制 NF-κB,Wnt,PI3K-Akt,MAPK 和 JAK-STAT 信号通路。它通过抑制NF-κB 而诱导肿瘤细胞凋亡。 | |||
TN5952 |
2,3-Dihydro-3α-methoxynimbolide
|
||
2,3-Dihydro-3α-methoxynimbolide induces apoptosis via both mitochondrial and death receptor pathways in stomach (AZ521) cancer cell line. | |||
TN2835 |
28-Deoxonimbolide
|
Caspase | Apoptosis; Proteases/Proteasome |
28-Deoxonimbolide exhibits potent cytotoxic activity against HL60 leukemia cells. |