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Search Results for " nematicidal "

3

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T21687 Conoidin A

Parasite Microbiology/Virology
Conoidin A 是刚地弓形虫过氧化物酶 II 的细胞通透性抑制剂,有杀线虫特性。它共价结合 TgPrxII 的过氧化物催化位点 Cys47,不可逆地抑制其过氧化物活性,IC50为 23 µM。它也抑制哺乳动物 PrxI 和 PrxII 的氧化。它具有抗氧化、神经保护作用,可研究缺血性心脏病。
T37673 Asperlactone

Asperlactone is a nematicidal, insecticidal, antibacterial, and antifungal polyketide metabolite produced from A. westerdijkiae.
T37674 Aspyrone

Aspyrone is a polyketide fungal metabolite that has been found inAspergillusand has diverse biological activities.1,2It is active against a panel of 13 fungi when used at a concentration of 20 μg/ml and a panel of 21 bacteria in a disc assay when used at a concentration of 100 μg per disc.1Aspyrone (10-1,000 mg/L) is nematocidal againstP. penetrans.2 1.Torres, M., Balcells, M., Sala, N., et al.Bactericidal and fungicidal activity of Aspergillus ochraceus metabolites and some derivativesPestic. S...

化合物

Conoidin A
Cat.No: T21687
Synonym:
Target: Parasite
Asperlactone
Cat.No: T37673
Synonym:
Target:
Aspyrone
Cat.No: T37674
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T15277 Fervenulin

Parasite Microbiology/Virology
Fervenulin 具有杀灭线虫活性,抑制线虫M. incognita 卵孵化和 J2 的校正死亡率,MIC 分别为 30 μg/mL 和 120 μg/mL。
TN1977 Neochamaejasmine B

新狼毒素B

Antifection Microbiology/Virology
Neochamaejasmin B 是一种提取自Stellera chamaejasme L.的双黄酮化合物。它在 C-2/C-3 和 C-2″/C-3″ 位置具有顺反几何结构。
T67670 4-Ethylbenzaldehyde

Endogenous Metabolite Metabolism
4-Ethylbenzaldehyde 是一种 RIFM 香料,存在于自然发酵的罗非鱼香肠和大豆植株中。4-Ethylbenzaldehyde 在250 g/ml 时显示出杀线虫活性,可被当作一种新型杀线虫剂。
TN1343 8-Geranyloxypsoralen

8-香叶草氧基补骨脂素

Anti-infection; P450; BACE Metabolism; Microbiology/Virology; Neuroscience
8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。
T3897 Isoschaftoside

Anti-infection; Antifungal Microbiology/Virology
Isoschaftosid 是从 Desmodium uncinatum 根部分泌物中提取的 c- 糖基黄酮类天然产物,有抗肿瘤、抗氧化和抗菌活性,它还对 M. incognita 具有很强的杀线虫活性。
TN3409 Anagyrine

Antifection Microbiology/Virology
Anagyrine, is the responsible teratogen from teratogenic lupins, can produce congenital deformities in calves typical of crooked calf disease; it also can induce red cell aplasia, vascular anomaly, and skeletal dysplasia.(-)-Anagyrine and (-)--Methylcytisine have nematicidal activities against Pine Wood Nematodes.
TN3112 5-Heneicosylresorcinol

NADPH-oxidase; Antifection Immunology/Inflammation; Microbiology/Virology
5-Heneicosylresorcinol 对 RBL-2H3 细胞中 β-己糖胺酶的释放具有抑制作用,它还可以防止 3T3-L1 细胞中甘油三酯的积累。它对红线虫、秀丽隐杆线虫和松材线虫具有杀线虫活性,ED50 值分别为 80、30 和 180 ug/mL。
TN3573 Camaric acid

Antifection Microbiology/Virology
Camaric acid shows antibacterial activity against Staphylococcus aureus and methicillin resistant S. aureus with IC50 values 8.74 and 8.09 uM, respectively, it also shows moderate antileishmanial activity and highly potent antitrypanosomal activity. Camar
T4S0083 Protostemonine

Others Others
Protostemonine 是一种主要从 Stemona sesslifolia 根中分离得到的生物碱,对哮喘及革兰氏阴性菌所致急性肺损伤有抗炎作用。

天然产物

Fervenulin
Cat.No: T15277
Synonym:
Target: Parasite
Neochamaejasmine B
Cat.No: TN1977
Synonym: 新狼毒素B
Target: Antifection
4-Ethylbenzaldehyde
Cat.No: T67670
Synonym:
Target: Endogenous Metabolite
8-Geranyloxypsoralen
Cat.No: TN1343
Synonym: 8-香叶草氧基补骨脂素
Target: Anti-infection, P450, BACE
Isoschaftoside
Cat.No: T3897
Synonym:
Target: Anti-infection, Antifungal
Anagyrine
Cat.No: TN3409
Synonym:
Target: Antifection
5-Heneicosylresorcinol
Cat.No: TN3112
Synonym:
Target: NADPH-oxidase, Antifection
Camaric acid
Cat.No: TN3573
Synonym:
Target: Antifection
Protostemonine
Cat.No: T4S0083
Synonym:
Target: Others
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