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Cat. No. Product Name Target Signaling Pathways
T23052 Nafamostat

Others Others
Nafamostat is a synthetic serine protease inhibitor and is an anticoagulant.
T2392 Nafamostat mesylate

甲磺酸萘莫司他,FUT-175

Apoptosis; Serine/threonin kinase; SARS-CoV; Serine Protease Apoptosis; Cell Cycle/Checkpoint; Metabolism; Microbiology/Virology; Proteases/Proteasome
Nafamostat mesylate (FUT-175) 是一种广谱丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固。它通过降低颗粒酶活性和 CTL 细胞溶解抑制T 细胞自身反应活性,可抑制SARS-CoV-2 的激活。它还是潜在的补体抑制剂。
T23051 Nafamostat hydrochloride

Others Others
Nafamostat hydrochloride is a synthetic serine protease inhibitor and is an anticoagulant.
T37096 Sepimostat dimethanesulfonate

Sepimostat dimethanesulfonate (FUT-187) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dimethanesulfonate inhibits the Ifenprodil binding with a Ki value of 27.7 μM[1]. Sepimostat (1 to 100 nmol/eye, intravitreal injection) exhibits significant neuroprotective effect[1]. ...

化合物

Nafamostat
Cat.No: T23052
Synonym:
Target: Others
Nafamostat mesylate
Cat.No: T2392
Synonym: 甲磺酸萘莫司他,FUT-175
Target: Apoptosis, Serine/threonin kinase, SARS-CoV, Serine Protease
Nafamostat hydrochloride
Cat.No: T23051
Synonym:
Target: Others
Sepimostat dimethanesulfonate
Cat.No: T37096
Synonym:
Target:
TargetMol Loading
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