Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1023 |
Miltirone
|
P450; GABA Receptor | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Miltirone 是存在于丹参中的一种天然产物,可作为中枢苯二氮受体部分激动剂,IC50值为 0.3 μM。 | |||
T83425 |
1-Oxomiltirone
|
||
2-Isopropyl-8,8-dimethyl-7,8-dihydrophenanthrene-3,4,5(6H)-trione 为C20-norabietane类二萜化合物,具备抗炎作用,可从鼠尾草叶中提取。 | |||
TN1562 |
Dehydromiltirone
|
NOS; NF-κB; COX | Immunology/Inflammation; Neuroscience; NF-κB |
Dehydromiltirone has antioxidant activity, it shows significant anti-neuroinflammatory effects through inhibiting PI3K/Akt phosphorylation and then inhibiting NF-κB signaling pathway. |