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Cat. No. Product Name Target Signaling Pathways
T76653 Polybia-MP1

Polybia-MP1 是一种抗菌素乳苦菌肽。
T80585 Anti-Mouse GM-CSF Antibody (MP1-22E9)

c-Fms Tyrosine Kinase/Adaptors
Anti-MouseGM-CSFAntibody 为特异性针对小鼠GM-CSF的IgG2a类免疫球蛋白抗体,由大鼠血清中提取。
T69977 BC-1485

BC-1485 is a first-in-class inhibitor of Fibrosis-inducing E3 ligase 1 (FIEL1 ), which disrupts FIEL1-directed PIAS4 ubiquitination.
T71901 MP-1

MP-1 is a covalent inhibitor of fumarate hydratase (FH) that exhibits cytotoxicity dependent on FH. MP-1 engages a functional cysteine in the Zn-finger domain of the tRNA methyltransferase enzyme TRMT1.
T16124 MMP13-IN-3

MMP Proteases/Proteasome
MMP13-IN-3 是口服有效的MMP-13选择性抑制剂,IC50为 1 nM,比其他 MMP 的选择性高 1000倍多。MMP13-IN-3在用于骨关节炎方面有研究的价值。
T3983 TMP195

TFMO 2,TMP 195

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
TMP195 (TFMO 2) 是一种选择性 IIa 类组蛋白脱乙酰酶 (HDAC) 抑制剂。对 HDAC4、HDAC5、HDAC7,HDAC9的 Ki 值分别为59、60、26,5 nM。
T78269 Anti-Mouse PD-1 Antibody (RMP1-14)

PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
RMP1-14 是一种 IgG1 样免疫球蛋白抗小鼠 PD-1 抗体,可阻断 PD-1/PD-L1 信号传导。
T41079 MMP13-IN-2

MMP13-IN-2

MMP13-IN-2 is a highly potent, selective, and orally active inhibitor of MMP-13. It demonstrates exceptional potency against MMP-13, with an IC50 value of 0.036 nM, and exhibits selectivities greater than 1,500-fold over MMP-1, 3, 7, 8, 9, 14, and TACE. Moreover, MMP13-IN-2 possesses the capability to effectively inhibit collagen release from cartilage in vitro. Consequently, MMP13-IN-2 holds great potential for advancing research on collagenase-related diseases.
T76244 Amp1EP9

Amp1EP9为一抗菌肽,作为开发有效无毒抗菌活性分子的强大工具,具备针对多重耐药细菌感染进行研究的潜力。
T80282 cPcAMP1/26

cPcAMP1/26 是一款抗菌肽,能高效清除A.Hydrophila及金黄色葡萄球菌 (S. aureus)。该化合物通过诱导细菌质膜去极化作用并提升细胞内ROS水平,展示其抗菌机制。
T78775 MMP13-IN-5

MMP Proteases/Proteasome
MMP13-IN-5 (compound 13m) 作为具有针对性的MMP-2/MMP-13 抑制剂,显示出高效的抑制活性(IC50=3.6 μM/14.6 μM),适用于骨关节炎疼痛的研究。
T83487 [Pmp1,Tyr(OEt)2] AVP

[Pmp1,Tyr(OEt)2] AVP为环状加压素(AVP)的线性拮抗剂,具备相似结构。
T78774 MMP13-IN-4

MMP Proteases/Proteasome
MMP13-IN-4(compound 13)作为MMP-13抑制剂,具备强效性和选择性,其IC50值为14.6 μM,可用于骨关节炎疼痛的研究。
T72306 Mycobacterial Zmp1-IN-1

Mycobacterial Zmp1-IN-1 是一种分枝杆菌锌金属蛋白酶-1(Zmp1)抑制剂。Mycobacterial Zmp1-IN-1 对 MtbH37Ra 具有剂量依赖性抑制的抗分枝杆菌活性。Mycobacterial Zmp1-IN-1 可用于结核病 (TB) 的研究。
T80336 DFTamP1

DFTamP1为抗菌肽,针对金黄色葡萄球菌USA300表现出活性,其最小抑菌浓度(MIC)为3.1 μM。
T82063 Integrin signaling inhibitor, mP13

Integrinsignaling inhibitor, mP13 是抑制整合素信号传导,阻止内向外和外向内信号传递,涉及纤维蛋白原结合、血小板粘附及凝块收缩的化合物。

化合物

Polybia-MP1
Cat.No: T76653
Synonym:
Target:
Anti-Mouse GM-CSF Antibody (MP1-22E9)
Cat.No: T80585
Synonym:
Target: c-Fms
BC-1485
Cat.No: T69977
Synonym:
Target:
MP-1
Cat.No: T71901
Synonym:
Target:
MMP13-IN-3
Cat.No: T16124
Synonym:
Target: MMP
TMP195
Cat.No: T3983
Synonym: TFMO 2,TMP 195
Target: HDAC
Anti-Mouse PD-1 Antibody (RMP1-14)
Cat.No: T78269
Synonym:
Target: PD-1/PD-L1
MMP13-IN-2
Cat.No: T41079
Synonym: MMP13-IN-2
Target:
Amp1EP9
Cat.No: T76244
Synonym:
Target:
cPcAMP1/26
Cat.No: T80282
Synonym:
Target:
MMP13-IN-5
Cat.No: T78775
Synonym:
Target: MMP
[Pmp1,Tyr(OEt)2] AVP
Cat.No: T83487
Synonym:
Target:
MMP13-IN-4
Cat.No: T78774
Synonym:
Target: MMP
Mycobacterial Zmp1-IN-1
Cat.No: T72306
Synonym:
Target:
DFTamP1
Cat.No: T80336
Synonym:
Target:
Integrin signaling inhibitor, mP13
Cat.No: T82063
Synonym:
Target:
TargetMol Loading
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