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Cat. No.	Product Name	Target	Signaling Pathways
T79060	MOR agonist-1	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	MOR agonist-1为一种针对MOR（μ-opioid receptor）的激动剂，展现出优秀的镇痛效果，适用于疼痛及其相关疾病的研究应用。
T79547	MOR agonist-2	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	MOR agonist-2 (Compound 46) 为D3R拮抗剂及MOR激动剂，其Ki值分别为7.26 nM和564 nM。MOR agonist-2潜在以MOR部分激动机制实现镇痛效果，并通过D3R拮抗降低阿片类药物的滥用风险。
T81763	MOR agonist-3
	MOR Agonist-3 (Compound 84) 是一种双重作用化合物，具有D3R/MOR拮抗活性（Ki值为55.2 nM和382 nM）。该化合物其MOR部分激动性质展现出镇痛潜力，并可能通通过D3R拮抗作用降低阿片类药物的滥用风险。MOR Agonist-3 亦适用于炎症治痈和神经性疼痛的研究领域。
T62268	μ opioid receptor agonist 1
	μ opioid receptor agonist 1 （Compound H-1a）是一种光学纯的氧杂环取代吡咯并吡唑衍生物，也是一种 MOR 受体激动剂，能够用于研究疼痛及疼痛相关疾病。
T9669	EST73502 hydrochloride
	EST73502 hydrochloride 是一种选择性的，具有口服活性和血脑屏障渗透性的 μ-opioid 受体 (μ-opioid receptor/MOR) 激动剂和 σ1 受体(σ1R) 拮抗剂，对 MOR 和 σ1R 作用的Ki 值分别为 64 nM 和 118 nM。EST73502 hydrochloride 可用于缓解疼痛研究。
T69537	Difelikefalin HCl
	Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin HCl is selective for KOR over the μ-opioid receptor (MOR; EC50 = >1 µM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07...
T37483	Difelikefalin (trifluoroacetate salt)
	Difelikefalin is a κ-opioid receptor (KOR) agonist.1It activates KOR in HEK293 cells expressing the human receptor (EC50= 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50= 0.048 nM). Difelikefalin is selective for KOR over the μ-opioid receptor (MOR; EC50= >1 μM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07 and 0.05 m...
T75916	Dynorphin A TFA
	Dynorphin A TFA, 作为一种内源性阿片肽，主要在中枢神经系统（CNS）中发挥抑制性神经传导的作用。该化合物不仅是kappa阿片受体（KOR）的高效激动剂，还能激活其他阿片受体，包括mu（MOR）和delta（DOR）。Dynorphin A TFA具有诱导神经元死亡的能力，因此在神经系统疾病的研究中具有应用价值。
T69530	Difelikefalin TFA
	Difelikefalin TFA is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin TFA is selective for KOR over the μ-opioid receptor (MOR; EC50 = >1 µM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07...