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Cat. No. Product Name Target Signaling Pathways
T8342 BRD9876

6-叔丁基-2,3-二氰基萘

Others; Kinesin; Microtubule Associated Cytoskeletal Signaling; Others
BRD9876 是一种 MM1S 生长的选择性抑制剂,可将驱动蛋白 5 锁定在增强微管结合的状态,从而导致 MT 的捆绑和稳定。它特异性靶向微管结合的 Eg5,选择性抑制 CD34 细胞的骨髓瘤,有用于多发性骨髓瘤的研究潜力。
T11751 KDOAM-25

Antibacterial Microbiology/Virology
KDOAM-25, a potent and highly selective inhibitor of histone lysine demethylases 5 (KDM5) with IC50 values of 71 nM for KDM5A, 19 nM for KDM5B, 69 nM for KDM5C, and 69 nM for KDM5D, enhances global H3K4 methylation at transcriptional start sites and reduces proliferation in multiple myeloma MM1S cells.
T11750L KDOAM-25 trihydrochloride (2230731-99-2 free base)

KDOAM-25 trihydrochloride

Others Others
KDOAM-25 trihydrochloride increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells. KDOAM-25 trihydrochloride is a potent and highly selective histone lysine demethylases 5 (KDM5) inhibitor
T11750 KDOAM-25 citrate

Others Others
KDOAM-25 citrate 是有效且具有高选择性的组蛋白赖氨酸脱甲基酶 5 (KDM5) 抑制剂,对 KDM5A,KDM5B,KDM5C,KDM5D 的IC50分别为 71 nM,19 nM,69 nM,69 nM。用KDOAM-25 citrate 处理的多发性骨髓瘤 MM1S 细胞显示转录起始位点的整体 H3K4 甲基化增加,增殖受损。
T35479 CRBN-6-5-5-VHL

Potent and selective cereblon degrader (DC50 = 1.5 nM). Induces complete degradation of cereblon in MM1S cells. Comprises a cereblon E3 ligase ligand joined by a linker to a ligand for the E3 ligase VHL. Cell-permeable. Steinebach et al (2019) PROTAC-mediated crosstalk between E3 ligases. Chem.Commun.(Camb) 55 1821 PMID:30672516
T62166 KDOAM-25 trihydrochloride

KDOAM-25 trihydrochloride 是一种有效的、高度选择性的组蛋白赖氨酸脱甲基酶 5 (KDM5) 抑制剂,能够作用于 KDM5A (IC50: 71 nM)、KDM5B (IC50: 19 nM)、KDM5C (IC50: 69 nM)、KDM5D (IC50: 69 nM)。KDOAM-25 trihydrochloride 能够提高转录起始位点的整体 H3K4 甲基化,可阻碍多发性骨髓瘤 MM1S 细胞的增殖。

化合物

BRD9876
Cat.No: T8342
Synonym: 6-叔丁基-2,3-二氰基萘
Target: Others, Kinesin, Microtubule Associated
KDOAM-25
Cat.No: T11751
Synonym:
Target: Antibacterial
KDOAM-25 trihydrochloride (2230731-99-2 free base)
Cat.No: T11750L
Synonym: KDOAM-25 trihydrochloride
Target: Others
KDOAM-25 citrate
Cat.No: T11750
Synonym:
Target: Others
CRBN-6-5-5-VHL
Cat.No: T35479
Synonym:
Target:
KDOAM-25 trihydrochloride
Cat.No: T62166
Synonym:
Target:
TargetMol Loading
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