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Cat. No. Product Name Target Signaling Pathways
T33451 ML 7

ML7,ML-7

ML 7 is an inhibitor of myosin light chain kinase that protects cardiac function from ischemia/reperfusion (I/R) injury.
T3050 ML-7 hydrochloride

ML-7 HCl,ML-7盐酸盐

Serine/threonin kinase; Myosin; YAP; PKA; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
ML-7 hydrochloride (ML-7 HCl) 是一种可渗透细胞的、可逆的、有效的、ATP 竞争性的肌球蛋白轻链激酶(MLCK) 特异性抑制剂,IC50为300 nM。它还抑制平滑肌肌球蛋白轻链激酶、PKA 和 PKC。
T11185 EML741

Histone Methyltransferase Chromatin/Epigenetic
EML741 also inhibits DNMT1 (IC50, 3.1 μM), with no effect on DNMT3a or DNMT3b. EML741 exhibits low cell toxicity, and is membrane permeable and blood-brain barrier penetrated. EML741 is a histone lysine methyltransferase G9a/GLP inhibitor, with an IC50 of 23 nM, Kd of 1.13 μM for G9a.
T16113 ML753286

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
ML753286 has high permeability and low to medium clearance in rodent and human liver S9 fractions. ML753286 is an orally active and selective inhibitor of BCRP (IC50: 0.6 μM). It is also stable in plasma across species.
T79614 EML734

Histone Methyltransferase Chromatin/Epigenetic
EML734为PRMT7/9的选择性抑制剂,其对PRMT7的IC50为315 nM,对PRMT9的IC50为0.89 μM。
T72861 (6R)-ML753286

(6R)-ML753286 是 ML753286 的异构体。ML753286 是一种口服活性和选择性 BCRP(抗乳腺癌蛋白) 抑制剂,IC50为 0.6 μM。 ML753286 在啮齿动物和人类肝脏 S9 组分中具有高渗透性和低至中等清除率,并且在不同物种中都具有血浆稳定性。
T10490 (S)-ML753286

Others Others
(S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).

化合物

ML 7
Cat.No: T33451
Synonym: ML7,ML-7
Target:
ML-7 hydrochloride
Cat.No: T3050
Synonym: ML-7 HCl,ML-7盐酸盐
Target: Serine/threonin kinase, Myosin, YAP, PKA, PKC
EML741
Cat.No: T11185
Synonym:
Target: Histone Methyltransferase
ML753286
Cat.No: T16113
Synonym:
Target: AMPK
EML734
Cat.No: T79614
Synonym:
Target: Histone Methyltransferase
(6R)-ML753286
Cat.No: T72861
Synonym:
Target:
(S)-ML753286
Cat.No: T10490
Synonym:
Target: Others
TargetMol Loading
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