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Cat. No. Product Name Target Signaling Pathways
T9034 MK2-IN-3

MK2 Inhibitor III

MAPK MAPK
MK2-IN-3 (MK2 Inhibitor III) 是选择性的 MAPKAP-K2 (MK-2)抑制剂(IC50:8.5 nM),能够抑制 U937 细胞及体内 TNFα 的生成。
T12058 MK2-IN-3 hydrate

MK-2 Inhibitor III

ERK; MAPK; MNK MAPK
MK2-IN-3 hydrate (MK-2 Inhibitor III) 是一种口服有活性的、ATP 竞争性的MAPKAP-K2 (MK-2)选择性抑制剂(IC50:0.85 nM)。
T81783 MK2-IN-5

Hsp25 kinase inhibitor,Mk2 pseudosubstrate

ERK MAPK
MK2-IN-5为Mk2的假底物,Ki值为8 μM。该化合物针对MAPK通路内的蛋白相互作用域,并能抑制HSP25与HSP27的磷酸化。
T35536 Tpl2 Kinase Inhibitor (hydrochloride)

Tpl2 kinase inhibitor is an inhibitor of tumor progression locus 2 (Tpl2; IC50= 0.05 μM).1It is selective for Tpl2 over MEK, p38 MAPK, Src, MK2, and PKC (IC50s = >40, 180, >400, 110, and >400 μM, respectively). Tpl2 kinase inhibitor inhibits LPS-induced TNF-α production in isolated human monocytes and whole blood (IC50s = 0.7 and 8.5 μM, respectively). It enhances differentiation induced by calcitriol in HL-60 and U937 leukemia cells when used at a concentration of 5 μM.2Tpl2 kinase inhibitor (5...

化合物

MK2-IN-3
Cat.No: T9034
Synonym: MK2 Inhibitor III
Target: MAPK
MK2-IN-3 hydrate
Cat.No: T12058
Synonym: MK-2 Inhibitor III
Target: ERK, MAPK, MNK
MK2-IN-5
Cat.No: T81783
Synonym: Hsp25 kinase inhibitor,Mk2 pseudosubstrate
Target: ERK
Tpl2 Kinase Inhibitor (hydrochloride)
Cat.No: T35536
Synonym:
Target:
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