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Cat. No. Product Name Target Signaling Pathways
T0242 Sitagliptin

西他列汀,MK0431,西格列汀

Proteasome; DPP-4; Autophagy Autophagy; Proteases/Proteasome; Ubiquitination
Sitagliptin (MK0431) 是一种有效的 DPP4抑制剂,在 Caco-2 细胞中,IC50值为 19 nM。它是一种新型口服降糖药,可单独使用或与二甲双胍或噻唑烷二酮联合用于治疗 2 型糖尿病。
T23358 Sitagliptin phosphate

磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)

DPP-4; Autophagy Autophagy; Proteases/Proteasome
Sitagliptin phosphate (MK-0431 phosphate) 是一种二肽基肽酶 4 (DPP4) 抑制剂,在 Caco-2 细胞中,IC50值为 19 nM。
T0242L Sitagliptin phosphate monohydrate

MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物

Proteasome; DPP-4; Autophagy Autophagy; Proteases/Proteasome; Ubiquitination
Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) 是一种有效的 DPP-IV 抑制剂,在 Caco-2 细胞提取物中的 IC50 为 19 nM。
T40930 (S)-Sitagliptin phosphate

(S)-Sitagliptin phosphate,(S)-MK-0431 phosphate

(S)-Sitagliptin phosphate, the less active S-enantiomer of Sitagliptin phosphate, is a high-potency inhibitor of DPP4. It exhibits an IC50 of 19 nM in Caco-2 cell extracts.

化合物

Sitagliptin
Cat.No: T0242
Synonym: 西他列汀,MK0431,西格列汀
Target: Proteasome, DPP-4, Autophagy
Sitagliptin phosphate
Cat.No: T23358
Synonym: 磷酸西他列汀,Januvia,MK-0431 phosphate,Sitagliptin (phosphate)
Target: DPP-4, Autophagy
Sitagliptin phosphate monohydrate
Cat.No: T0242L
Synonym: MK-0431,MK-0431 phosphate monohydrate,西他列汀磷酸盐一水合物
Target: Proteasome, DPP-4, Autophagy
(S)-Sitagliptin phosphate
Cat.No: T40930
Synonym: (S)-Sitagliptin phosphate,(S)-MK-0431 phosphate
Target:
TargetMol Loading
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