Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2379 |
UNC1215
|
Apoptosis; Epigenetic Reader Domain; Histone Methyltransferase | Apoptosis; Chromatin/Epigenetic |
UNC1215 是一种选择性 L3MBTL3甲基赖氨酸结构域的拮抗剂,IC50为40 nM,Kd 为 120 nM。它可研究恶性脑瘤。 | |||
T2252 |
UNC 669
UNC669 |
Epigenetic Reader Domain | Chromatin/Epigenetic |
UNC 669是一种有效且特异性的 MBT(恶性脑瘤)抑制剂,是甲基赖氨酸结合结构域的配体,是L3MBTL1和L3MBTL3的抑制剂,IC50分别为 4.2 和 3.1 uM。 | |||
T71101 | DMBT | ||
DMBT is an inhibitor of invasion and metastasis through Akt/GSK-3β/β-catenin pathway in B16BL6 cells. |