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Cat. No. Product Name Target Signaling Pathways
T21337 Lurasidone

SM-13496,鲁拉西酮

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Lurasidone (SM-13496) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。
T1735 Lurasidone hydrochloride

Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496

Dopamine Receptor; 5-HT Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。
T11893L Lurasidone metabolite 14326 hydrochloride

Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base)

Others Others
Lurasidone metabolite 14326 hydrochloride, an active metabolite of the atypical antipsychotic Lurasidone, maintains its significant function in pharmacological efficacy.
T11893 Lurasidone metabolite 14326

Others Others
Lurasidone metabolite 14326, an active metabolite of the atypical antipsychotic Lurasidone, functions effectively in the body.
T11892 Lurasidone D8 Hydrochloride

SM-13496 D8

Others Others
Lurasidone D8 Hydrochloride is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone.
T19406 Lurasidone Metabolite 14283 D8

Others Others
Lurasidone Metabolite 14283 D8 is the deuterium labeled Lurasidone Metabolite 14283.
T19407 Lurasidone Metabolite 14326 D8

Others Others
Lurasidone Metabolite 14326 D8 is the deuterium labeled Lurasidone Metabolite 14326.
T13760 Lurasidone Metabolite 14283 hydrochloride

Others Others
Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone.

化合物

Lurasidone
Cat.No: T21337
Synonym: SM-13496,鲁拉西酮
Target: Dopamine Receptor, 5-HT Receptor
Lurasidone hydrochloride
Cat.No: T1735
Synonym: Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine
Lurasidone metabolite 14326 hydrochloride
Cat.No: T11893L
Synonym: Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base)
Target: Others
Lurasidone metabolite 14326
Cat.No: T11893
Synonym:
Target: Others
Lurasidone D8 Hydrochloride
Cat.No: T11892
Synonym: SM-13496 D8
Target: Others
Lurasidone Metabolite 14283 D8
Cat.No: T19406
Synonym:
Target: Others
Lurasidone Metabolite 14326 D8
Cat.No: T19407
Synonym:
Target: Others
Lurasidone Metabolite 14283 hydrochloride
Cat.No: T13760
Synonym:
Target: Others
TargetMol Loading
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