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4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T37647 5α-dihydro Levonorgestrel

5α-dihydro Levonorgestrel is a metabolite of the synthetic progestin levonorgestrel . It lacks in vitro and in vivo estrogenic activity, but induces copulatory behavior in male rats when administered at a dose of 1 mg per animal per day.
T32713 Levonorgestrel hexanoate

Plan B

Levonorgestrel hexanoate is a manufactured hormone used in a number of birth control methods.
T31699 Ethinylestradiol mixture with Levonorgestrel

Ethinylestradiol mixture with Levonorgestrel is formulated with increasing dosages of levonorgestrel and ethinyl estradiol.
T32712 Levonorgestrel butyrate

Levonorgestrel butyrate is a manufactured hormone used in a number of birth control methods.

化合物

5α-dihydro Levonorgestrel
Cat.No: T37647
Synonym:
Target:
Levonorgestrel hexanoate
Cat.No: T32713
Synonym: Plan B
Target:
Ethinylestradiol mixture with Levonorgestrel
Cat.No: T31699
Synonym:
Target:
Levonorgestrel butyrate
Cat.No: T32712
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T7044 Norepinephrine

去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol

MMP; Endogenous Metabolite; Adrenergic Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Neuroscience; Proteases/Proteasome
Norepinephrine (Levophed) 是β1选择性的肾上腺素能受体激动剂,EC50值为 5.37 μM。它可上调鼻咽癌肿瘤细胞中血管内皮生长因子、基质金属蛋白酶MMP-2和MMP-9的表达。
T1263 Levonorgestrel

左炔诺孕酮,D-Norgestrel

Others; Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Levonorgestrel (D-Norgestrel) 是一种合成孕激素,可作用于孕酮受体。它是一种宫内节育器,可以抑制卵子受精。

天然产物

Norepinephrine
Cat.No: T7044
Synonym: 去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol
Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy
Levonorgestrel
Cat.No: T1263
Synonym: 左炔诺孕酮,D-Norgestrel
Target: Others, Estrogen/progestogen Receptor, Progesterone Receptor
TargetMol Loading
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