Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1876 |
Kobe0065
|
Apoptosis; Raf; Ras | Apoptosis; GPCR/G Protein; MAPK |
Kobe0065 是一种新型 Ras-Raf 相互作用抑制剂,可完全抑制 H-Ras·GTP 与 c-Raf-1 RBD 的结合,Ki 值为 46±13 μM。 | |||
T24267 |
Kobe2601
Kobe 2601,Kobe-2601 |
||
Kobe2601 is a Kobe0065 and Kobe02602 water-soluble analog. It displays inhibitory activity towards Ras-Raf binding. |