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4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22450 Tyrphostin B44, (+) enantiomer

酪氨酸磷酸化抑制剂AG 835

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Tyrphostin B44, (+) enantiomer 是一种表皮生长因子受体 (EGFR) 激酶抑制剂,IC50 为 0.86 μM,活性低于 (-) 对映体。
T6721 Vinblastine

Microtubule Associated; AChR Cytoskeletal Signaling; Neuroscience
Vinblastine 抑制微管形成并抑制 nAChR 活性,IC50 为 8.9 μM,用于治疗某些类型的癌症。
T29434 4-Desacetylvinblastine hydrazide

DAVLBH,Deacetylvinblastine hydrazide,Desacetylvinblastine hydrazide

Deacetylvinblastine hydrazide, a cytotoxic vinca alkaloid often conjugated with folic acid to produce EC145, a novel folate-receptor targeted agent.
T18330 MC-Val-Cit-PAB-vinblastine

Others Others
MC-Val-Cit-PAB-vinblastine is a potent antitumor drug-linker conjugate for Antibody-Drug Conjugates (ADC), featuring vinblastine (a microtubule protein inhibitor) connected through the MC-Val-Cit-PAB ADC linker.

化合物

Tyrphostin B44, (+) enantiomer
Cat.No: T22450
Synonym: 酪氨酸磷酸化抑制剂AG 835
Target: EGFR
Vinblastine
Cat.No: T6721
Synonym:
Target: Microtubule Associated, AChR
4-Desacetylvinblastine hydrazide
Cat.No: T29434
Synonym: DAVLBH,Deacetylvinblastine hydrazide,Desacetylvinblastine hydrazide
Target:
MC-Val-Cit-PAB-vinblastine
Cat.No: T18330
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1668 Vinblastine sulfate

硫酸长春碱,NSC49842,Vincaleukoblastine sulfate salt

Microtubule Associated; AChR; Autophagy Autophagy; Cytoskeletal Signaling; Neuroscience
Vinblastine sulfate (Vincaleukoblastine sulfate salt) 是对各种癌症类型有细胞毒性的生物碱。 它可以抑制微管的形成,也可以抑制 nAChR,IC50值为8.9 μM。
T3022 Anhydrovinblastine

脱水长春碱,3',4'-Anhydrovinblastine

Others Others
3',4'-Anhydrovinblastine (3',4'-Anhydrovinblastine) 是一种提取自Catharanthus roseus 叶片的单萜吲哚生物碱。

天然产物

Vinblastine sulfate
Cat.No: T1668
Synonym: 硫酸长春碱,NSC49842,Vincaleukoblastine sulfate salt
Target: Microtubule Associated, AChR, Autophagy
Anhydrovinblastine
Cat.No: T3022
Synonym: 脱水长春碱,3',4'-Anhydrovinblastine
Target: Others
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