Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2146 |
Fulvestrant
氟维司群,ZM 182780,ZD 9238,ICI 182780 |
Apoptosis; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Autophagy | Apoptosis; Autophagy; Endocrinology/Hormones |
Fulvestrant (ZM 182780) 是一种雌激素受体 (ER) 拮抗剂 (IC50=9.4 nM),也是一种 GPR30 的激动剂。Fulvestrant 具有抗肿瘤活性,可以抑制细胞增殖,诱导细胞凋亡和自噬。 | |||
T71710 |
Fulvestrant sulfone
|
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Fulvestrant sulfone is a synthetic estrogen receptor antagonist. | |||
T11334 |
Fulvestrant (R enantiomer)
ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer |
Others | Others |
Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. | |||
T11335 |
Fulvestrant (S enantiomer)
ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer |
Others | Others |
Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. |