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Cat. No. Product Name Target Signaling Pathways
T6113 ICG-001

Apoptosis; Epigenetic Reader Domain; Wnt/beta-catenin Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Stem Cells
ICG001 是β-catenin/TCF 介导的一种转录抑制剂,选择性地阻断 β-catenin/CBP 相互作用而不干扰 β-catenin/p300 相互作用。它可特异性结合 CREB 蛋白,IC50为3 μM。
T2237 ICG001

Epigenetic Reader Domain; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; Stem Cells
ICG001 (PRI-724 isomer) 拮抗 Wnt/β-catenin/TCF 介导的转录,并特异性结合元件结合蛋白(CREB) 结合蛋白 (CBP),IC50 为 3 μM,但不是相关的转录共激活因子 p300。
T64414 PRI-724

C-82 prodrug,Foscenvivint

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
PRI-724 (C-82 prodrug)是β-catenin/CBP 相互作用的选择性小分子抑制剂。
T65994 (6S)-N-Benzyl-6-(4-hydroxybenzyl)-8-(naphthalen-1-ylmethyl)-4,7-dioxohexahydro-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide

Wnt signaling is required for direct multiple biological processes and also plays key roles in the pathogenesis of various diseases. Cyclic AMP response element-binding protein (CREB) is a transcription factor that is a member of the leucine zipper family of DNA binding proteins. This protein binds as a homodimer to the cAMP-responsive element, an octameric palindrome. The protein is phosphorylated by several protein kinases, and induces transcription of genes in response to hormonal stimulation...

化合物

ICG-001
Cat.No: T6113
Synonym:
Target: Apoptosis, Epigenetic Reader Domain, Wnt/beta-catenin
ICG001
Cat.No: T2237
Synonym:
Target: Epigenetic Reader Domain, Wnt/beta-catenin
PRI-724
Cat.No: T64414
Synonym: C-82 prodrug,Foscenvivint
Target: Wnt/beta-catenin
(6S)-N-Benzyl-6-(4-hydroxybenzyl)-8-(naphthalen-1-ylmethyl)-4,7-dioxohexahydro-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide
Cat.No: T65994
Synonym:
Target:
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