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Cat. No. Product Name Target Signaling Pathways
T82176 HR1

HR1是一种乳突蛋白酶,可增加人红细胞膜渗透性,并能诱导细菌细胞质膜和肥大细胞质膜透化。
T11966 MCHR1 antagonist 2

HER; Melanin-concentrating Hormone Receptor (MCHR) Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors
MCHR1 antagonist 2 是有效的黑色素聚集激素受体 1 拮抗剂,IC50为 65 nM。它也抑制hERG,在IMR-32 细胞中的IC50为 4.0 nM。
T68796 Thr101

Thr101, also known as NOX Inhibitor VII, is a dose-dependent inhibitor of HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, and HDAC9. Thr101 is also a NOX inhibitor.
T11965 MCHR1 antagonist 3

Others Others
MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.
T10173 MCHR1 antagonist 1

Others Others
MCHR1 antagonist 1 is a selective antagonist of melanin-concentrating hormone-1 (MCH1) receptor (Kb: 1 nM, Ki: 4 nM at human MCH1).
T12904 SHR1653

Others Others
SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).
T39960 SHR168442

SHR168442

SHR168442 is a potent RORγ modulator, exhibiting an IC50 value of 0.035 μM.
T76270 SARS-CoV-2-IN-34

SARS-CoV-2-IN-34 (S-20-1) 是一种可穿透血脑屏障的 pan-coronavirus (CoV) fusion 抑制剂,具有广谱抑制活性。它能有效抑制伪型和真型 SARS-CoV-2 以及其变体 (VOCs) 的感染。SARS-CoV-2-IN-34 对 SARS-CoV-2 的 S1 和 S2 蛋白中的 HR1 和 RBD 结构域显示出高度亲和性,适用于感染研究。

化合物

HR1
Cat.No: T82176
Synonym:
Target:
MCHR1 antagonist 2
Cat.No: T11966
Synonym:
Target: HER, Melanin-concentrating Hormone Receptor (MCHR)
Thr101
Cat.No: T68796
Synonym:
Target:
MCHR1 antagonist 3
Cat.No: T11965
Synonym:
Target: Others
MCHR1 antagonist 1
Cat.No: T10173
Synonym:
Target: Others
SHR1653
Cat.No: T12904
Synonym:
Target: Others
SHR168442
Cat.No: T39960
Synonym: SHR168442
Target:
SARS-CoV-2-IN-34
Cat.No: T76270
Synonym:
Target:
TargetMol Loading
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