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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9597 |
H2S Donor 5a
N-(苯甲酰基硫基)苯甲酰胺 |
Endogenous Metabolite | Metabolism |
H2S Donor 5a 是一种稳定的、半胱氨酸活化的的 H2S 供体。它是研究 H2S 的有用工具。 | |||
T22830 |
GYY4137
GYY 4137 morpholine salt |
Others | Others |
GYY4137 (GYY 4137 morpholine salt) 是一种缓释H2S 供体,具有抗炎和抗癌作用,也具有血管扩张和抗高血压活性。 | |||
T3560 |
Desmethylanethol trithione
ADT-OH |
VEGFR; Akt | Angiogenesis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
Desmethylanethol trithione (ADT-OH) 是合成硫化氢的供体。它利用上调 FADD 诱导细胞凋亡,并对体内黑色素瘤的形成具有一定的抑制作用,可用于研究癌症疾病。 | |||
T36503 |
Sodium Hydrogen Sulfide (hydrate)
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Others | Others |
Sodium Hydrogen Sulfide (hydrate) 与一氧化氮一样,是一种重要的气体介质,对哺乳动物的免疫、神经、心血管和肺系统有重要影响。Sodium Hydrogen Sulfide (hydrate)是一种H2S 供体,常用于细胞和整个动物实验系统。例如,它被用来证明H2S 促进中性粒细胞迁移,减少气道炎症,保护神经轴突、心脏和肠道免受化学或缺血再灌注损伤。 | |||
T32293 |
JK-2 lithium
JK-2,JK2,JK 2 |
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JK-2 is a hydrogen sulfide (H2S) donor. At acidic pH, it shows a greatly accelerated H2S release upon protonation-induced intramolecular cyclization. | |||
T15361 | FW1256 | Others | Others |
FW1256 is a phenyl analog. It also a slow-releasing hydrogen sulfide (H2S) donor. FW1256 inhibits NF-κB activity and causes cell apoptosis. FW1256 shows potent anti-inflammatory effects. It also has the potential for cancer and cardiovascular disease trea | |||
T81396 |
PRO-F
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PRO-F是一种光活化H2S供体,具备ROS清除功能。该化合物通过光激活能生成荧光信号,实现H2S释放的实时追踪;其激活过程不耗费内源性成分。PRO-F在细胞内提供H2S,以防止ROS过量造成的细胞损害,并已在慢性伤口愈合和糖尿病模型中展现出促进效果。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8693 |
Diallyl Trisulfide
二烯丙基三硫化物,二烯丙基三硫醚 |
Apoptosis; Reactive Oxygen Species; Antifungal | Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Diallyl Trisulfide 是一种在大蒜中发现的有机多硫化物,可作为 H2S 供体。它抑制扩张性青霉的生长,有抗癌能力。 |