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Cat. No. Product Name Target Signaling Pathways
T11366 Garcinol

Apoptosis; Endogenous Metabolite; Histone Acetyltransferase; AChR; AChE Apoptosis; Chromatin/Epigenetic; Metabolism; Neuroscience
Garcinol 是一种从印度藤黄提取的聚异戊二烯基二苯甲酮,对乙酰胆碱酯酶和丁酰胆碱酯酶具有抗胆碱酯酶的特性,IC50分别为 0.66 µM 和 7.39 µM。它还抑制组蛋白乙酰转移酶和 p300/CPB 相关因子,具有抗炎和抗癌活性。
T75609 7-epi-Isogarcinol

7-epi-Isogarcinol 是一种PPAP(多环聚异戊二烯酰基间苯三酚),显示出适度的抗增殖活性。它通过阻断STAT3信号通路,诱导apoptosis(细胞凋亡)并抑制细胞迁移作用。
T36845 Isogarcinol

Isogarcinol is a natural polyisoprenylated benzophenone first isolated from plant species in the genus Garcinia. It has immunosuppressant actions, inhibiting the protein phosphatase calcineurin (IC50 = 36 μM) and suppressing the proliferation of T cells. Oral administration of isogarcinol in mice decreases delayed type hypersensitivity, prolongs graft survival in allogeneic skin transplants, suppresses inflammation in collagen-induced arthritis, and reduces clinical symptoms in experimental auto...

天然产物

Garcinol
Cat.No: T11366
Synonym:
Target: Apoptosis, Endogenous Metabolite, Histone Acetyltransferase, AChR, AChE
7-epi-Isogarcinol
Cat.No: T75609
Synonym:
Target:
Isogarcinol
Cat.No: T36845
Synonym:
Target:
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