Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6129 |
GSK-1070916
GSK-1070916A,GSK1070916 |
Apoptosis; Tie-2; FLT; AMPK; Aurora Kinase | Angiogenesis; Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
GSK-1070916 (GSK-1070916A) 是一种选择性,ATP 竞争型的极光激酶B/C 抑制剂,Ki 值分别为0.38和1.5 nM。 |