Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1817 |
GNF-2
GNF2 |
SARS-CoV; Bcr-Abl | Angiogenesis; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
GNF-2 是一种高选择性的非 ATP 竞争性 Bcr-Abl 抑制剂。 它抑制 Ba/F3.p210 增殖,IC50为 138 nM。 | |||
T1803 |
GNF-5
GNF 5 |
SARS-CoV; Bcr-Abl | Angiogenesis; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
GNF-5是 Bcr-Abl 的特异性非 ATP 竞争性抑制剂,IC50为0.22uM。它是 GNF-2 的类似物,具有改进的药代动力学特性。 | |||
T18996 |
GNF-2-PEG-acid
|
Others | Others |
GNF-2-PEG-acid is usually used as a fluorescent probe. | |||
T18593 |
GNF5-amido-Me
PROTAC ABL binding moiety 2 |
Others | Others |
GNF5-amido-Me, the moiety based on GNF5 (ABL inhibitor),binds through a linker to the IAP ligand forming SNIPER[1]. | |||
T10199 |
GNF-PF-3777
8-Nitrotryptanthrin |
IDO; Indoleamine 2,3-Dioxygenase (IDO) | Metabolism |
GNF-PF-3777 (8-Nitrotryptanthrin) 是人吲哚胺2,3-双加氧酶 2 (hIDO2) 抑制剂,能够降低IDO2活性,Ki=为 0.97 μM。 |