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Cat. No. Product Name Target Signaling Pathways
T2146 Fulvestrant

氟维司群,ZM 182780,ZD 9238,ICI 182780

Apoptosis; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones
Fulvestrant (ZM 182780) 是一种雌激素受体 (ER) 拮抗剂 (IC50=9.4 nM),也是一种 GPR30 的激动剂。Fulvestrant 具有抗肿瘤活性,可以抑制细胞增殖,诱导细胞凋亡和自噬。
T11334 Fulvestrant (R enantiomer)

ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer

Others Others
Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T11335 Fulvestrant (S enantiomer)

ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer

Others Others
Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T71710 Fulvestrant sulfone

Fulvestrant sulfone is a synthetic estrogen receptor antagonist.
T82366 Fulvestrant 3-β-D-Glucuronide

Fulvestrant 3-β-D-Glucuronide,Fulvestrant的代谢产物,为葡萄糖醛酸结合物,属于纯抗雌激素类固醇。该化合物可应用于乳腺癌研究领域。
T71578 Endoxifen mesylate

Endoxifen, also known as N-desmethyl-4-hydroxytamoxifen, is a chemical that is under development for estrogen receptor-positive breast cancer. It is also being evaluated as an antipsychotic for treatment of mania and other psychotic disorders. Endoxifen is a nonsteroidal selective estrogen receptor modulator (SERM) of the triphenylethylene group. It is an active metabolite of tamoxifen and has been found to be effective in patients that have failed previous hormonal therapies (tamoxifen, aromat...

化合物

Fulvestrant
Cat.No: T2146
Synonym: 氟维司群,ZM 182780,ZD 9238,ICI 182780
Target: Apoptosis, Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
Fulvestrant (R enantiomer)
Cat.No: T11334
Synonym: ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer
Target: Others
Fulvestrant (S enantiomer)
Cat.No: T11335
Synonym: ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer
Target: Others
Fulvestrant sulfone
Cat.No: T71710
Synonym:
Target:
Fulvestrant 3-β-D-Glucuronide
Cat.No: T82366
Synonym:
Target:
Endoxifen mesylate
Cat.No: T71578
Synonym:
Target:
TargetMol Loading
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