Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28531 |
Facinicline hydrochloride
RG3487 |
5-HT Receptor; AChR | GPCR/G Protein; Neuroscience |
Facinicline hydrochloride (RG3487) 是一种口服有效的烟碱α7 receptor 部分激动剂,对人 nAChR 的 Ki 值为 6 nM。它可改善啮齿类动物的认知和感觉运动门控。它与5-HT3受体结合的 Ki 为 1.2 nM。 | |||
T31741 |
Facinicline (free base)
MEM-3454,RO-5313534,RG-3487,RG3487,R-3487,Facinicline |
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Facinicline (free base) is a partial agonist of the nicotinic alpha-7 (α7) receptor. It is used for the oral treatment of Alzheimer's. |